Compile Data Set for Download or QSAR
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Found 15 Enz. Inhib. hit(s) with all data for entry = 1374
TargetNADPH oxidase 4(Homo sapiens (Human))
Glucox Biotech

US Patent
LigandPNGBDBM318940(US10173988, Compound inventive)
Affinity DataIC50:  670nMAssay Description:Cells: HEK (CJ Nox4) stably expressing Nox4 was purchased from Redoxis AB (Lund). The adherent cells were cultivated in RPMI 1640 with L-Glutamine we...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNADPH oxidase 4(Homo sapiens (Human))
Glucox Biotech

US Patent
LigandPNGBDBM318937(US10173988, Compound B)
Affinity DataIC50:  840nMAssay Description:Cells: HEK (CJ Nox4) stably expressing Nox4 was purchased from Redoxis AB (Lund). The adherent cells were cultivated in RPMI 1640 with L-Glutamine we...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCytochrome b-245 heavy chain(Homo sapiens (Human))
Glucox Biotech

US Patent
LigandPNGBDBM318936(US10173988, Compound A)
Affinity DataIC50:  1.68E+3nMAssay Description:Cells: Human blood was purchased in buffy coat, prepared the same day for isolation of neutrophils, from Labjoy AB, Lund, Sweden. Blood components we...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNADPH oxidase 4(Homo sapiens (Human))
Glucox Biotech

US Patent
LigandPNGBDBM318936(US10173988, Compound A)
Affinity DataIC50:  1.68E+3nMAssay Description:Cells: HEK (CJ Nox4) stably expressing Nox4 was purchased from Redoxis AB (Lund). The adherent cells were cultivated in RPMI 1640 with L-Glutamine we...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNADPH oxidase 4(Homo sapiens (Human))
Glucox Biotech

US Patent
LigandPNGBDBM318939(US10173988, Compound D)
Affinity DataIC50:  1.68E+3nMAssay Description:Cells: HEK (CJ Nox4) stably expressing Nox4 was purchased from Redoxis AB (Lund). The adherent cells were cultivated in RPMI 1640 with L-Glutamine we...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNADPH oxidase 4(Homo sapiens (Human))
Glucox Biotech

US Patent
LigandPNGBDBM318938(US10173988, Compound C)
Affinity DataIC50:  1.68E+3nMAssay Description:Cells: HEK (CJ Nox4) stably expressing Nox4 was purchased from Redoxis AB (Lund). The adherent cells were cultivated in RPMI 1640 with L-Glutamine we...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCytochrome b-245 heavy chain(Homo sapiens (Human))
Glucox Biotech

US Patent
LigandPNGBDBM318939(US10173988, Compound D)
Affinity DataIC50:  1.50E+4nMAssay Description:Cells: Human blood was purchased in buffy coat, prepared the same day for isolation of neutrophils, from Labjoy AB, Lund, Sweden. Blood components we...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCytochrome b-245 heavy chain(Homo sapiens (Human))
Glucox Biotech

US Patent
LigandPNGBDBM318940(US10173988, Compound inventive)
Affinity DataIC50:  1.60E+4nMAssay Description:Cells: Human blood was purchased in buffy coat, prepared the same day for isolation of neutrophils, from Labjoy AB, Lund, Sweden. Blood components we...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCytochrome b-245 heavy chain(Homo sapiens (Human))
Glucox Biotech

US Patent
LigandPNGBDBM318937(US10173988, Compound B)
Affinity DataIC50:  1.70E+4nMAssay Description:Cells: Human blood was purchased in buffy coat, prepared the same day for isolation of neutrophils, from Labjoy AB, Lund, Sweden. Blood components we...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNADPH oxidase 1(Homo sapiens (Human))
Glucox Biotech

US Patent
LigandPNGBDBM318937(US10173988, Compound B)
Affinity DataIC50:  2.20E+4nMAssay Description:CHO cells modified to stably express human Nox1 were grown in DMEM/F12 gibco 31331 containing 10% FBS and 1% pen/strep at 37° C. in air with 5% CO2. ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCytochrome b-245 heavy chain(Homo sapiens (Human))
Glucox Biotech

US Patent
LigandPNGBDBM318938(US10173988, Compound C)
Affinity DataIC50:  5.90E+4nMAssay Description:Cells: Human blood was purchased in buffy coat, prepared the same day for isolation of neutrophils, from Labjoy AB, Lund, Sweden. Blood components we...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNADPH oxidase 1(Homo sapiens (Human))
Glucox Biotech

US Patent
LigandPNGBDBM318940(US10173988, Compound inventive)
Affinity DataIC50:  6.60E+4nMAssay Description:CHO cells modified to stably express human Nox1 were grown in DMEM/F12 gibco 31331 containing 10% FBS and 1% pen/strep at 37° C. in air with 5% CO2. ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNADPH oxidase 1(Homo sapiens (Human))
Glucox Biotech

US Patent
LigandPNGBDBM318936(US10173988, Compound A)
Affinity DataIC50:  6.60E+4nMAssay Description:CHO cells modified to stably express human Nox1 were grown in DMEM/F12 gibco 31331 containing 10% FBS and 1% pen/strep at 37° C. in air with 5% CO2. ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetNADPH oxidase 1(Homo sapiens (Human))
Glucox Biotech

US Patent
LigandPNGBDBM318938(US10173988, Compound C)
Affinity DataIC50:  1.62E+5nMAssay Description:CHO cells modified to stably express human Nox1 were grown in DMEM/F12 gibco 31331 containing 10% FBS and 1% pen/strep at 37° C. in air with 5% CO2. ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNADPH oxidase 1(Homo sapiens (Human))
Glucox Biotech

US Patent
LigandPNGBDBM318939(US10173988, Compound D)
Affinity DataIC50:  2.00E+5nMAssay Description:CHO cells modified to stably express human Nox1 were grown in DMEM/F12 gibco 31331 containing 10% FBS and 1% pen/strep at 37° C. in air with 5% CO2. ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent