Compile Data Set for Download or QSAR
maximum 50k data
Found 234 Enz. Inhib. hit(s) with all data for entry = 1400
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320544(US10174035, Compound 87 | [5-(1,3-Dimethyl-1H-pyra...)
Affinity DataIC50:  3nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320553(US10174035, Compound 96 | [5-(1,3-Dimethyl-1H-pyra...)
Affinity DataIC50:  3nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320554(US10174035, Compound 97 | [4-(Dimethylamino)piperi...)
Affinity DataIC50:  3nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320591(US10174035, Compound 134 | [4-(Morpholin-4-yl)pipe...)
Affinity DataIC50:  3nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320544(US10174035, Compound 87 | [5-(1,3-Dimethyl-1H-pyra...)
Affinity DataIC50:  3nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320554(US10174035, Compound 97 | [4-(Dimethylamino)piperi...)
Affinity DataIC50:  3nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320551(US10174035, Compound 94 | [5-(1,3-Dimethyl-1H-pyra...)
Affinity DataIC50:  4nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320551(US10174035, Compound 94 | [5-(1,3-Dimethyl-1H-pyra...)
Affinity DataIC50:  4nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320580(US10174035, Compound 123 | {6-Fluoro-7-(morpholin-...)
Affinity DataIC50:  4nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320576(US10174035, Compound 119 | {3-[(2R,6S)-2,6-dimethy...)
Affinity DataIC50:  5nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320541(US10174035, Compound 84 | [5-(1,3-Dimethyl-1H-pyra...)
Affinity DataIC50:  5nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320555(US10174035, Compound 98 | [6-Fluoro-5-(1-methyl-1H...)
Affinity DataIC50:  6nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320570(US10174035, Compound 113 | {4-[cis-2,6-Dimethylmor...)
Affinity DataIC50:  6nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320555(US10174035, Compound 98 | [6-Fluoro-5-(1-methyl-1H...)
Affinity DataIC50:  6nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320570(US10174035, Compound 113 | {4-[cis-2,6-Dimethylmor...)
Affinity DataIC50:  6nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320537(US10174035, Compound 81 | [6-Fluoro-5-(1-methyl-1H...)
Affinity DataIC50:  7nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320529(4-(1-{[6-(Morpholin-4-yl)-2-(1H-pyrazol-4-yl)-9H-p...)
Affinity DataIC50:  8nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320532(4-(1-{[5-(1-Methyl-1H-pyrazol-4-yl)-7-(morpholin-4...)
Affinity DataIC50:  9nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320496(US10174035, Compound 42 | [4-(Morpholin-4-yl)piper...)
Affinity DataIC50:  9nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320462(US10174035, Compound 9 | [2-(1,3-Dimethyl-1H-pyraz...)
Affinity DataIC50:  9nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320577(US10174035, Compound 120 | [5-(1-Methyl-1H-pyrazol...)
Affinity DataIC50:  10nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320586(1-Methyl-4-(1-{[5-(1-methyl-1H-pyrazol-4-yl)-7-(mo...)
Affinity DataIC50:  10nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320461(2-(4-{[2-(1,3-Dimethyl-1H-pyrazol-4-yl)-6-(morphol...)
Affinity DataIC50:  10nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320461(2-(4-{[2-(1,3-Dimethyl-1H-pyrazol-4-yl)-6-(morphol...)
Affinity DataIC50:  10nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320587(1-Methyl-4-(1-{[2-(1-methyl-1H-pyrazol-4-yl)-6-(mo...)
Affinity DataIC50:  10nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320521(9-Methyl-2-(1-methyl-1H-pyrazol-4-yl)-6-(morpholin...)
Affinity DataIC50:  11nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320538(2-(4-{[6-Fluoro-5-(1-methyl-1H-pyrazol-4-yl)-7-(mo...)
Affinity DataIC50:  11nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320458(US10174035, Compound 5 | {4-[cis-2,6-Dimethylmorph...)
Affinity DataIC50:  11nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320521(9-Methyl-2-(1-methyl-1H-pyrazol-4-yl)-6-(morpholin...)
Affinity DataIC50:  11nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320538(2-(4-{[6-Fluoro-5-(1-methyl-1H-pyrazol-4-yl)-7-(mo...)
Affinity DataIC50:  11nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320458(US10174035, Compound 5 | {4-[cis-2,6-Dimethylmorph...)
Affinity DataIC50:  11nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320519(US10174035, Compound 65 | {4-[cis-2,6-Dimethylmorp...)
Affinity DataIC50:  12nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320471(US10174035, Compound 17 | {2-[1-Methyl-3-(trifluor...)
Affinity DataIC50:  12nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320519(US10174035, Compound 65 | {4-[cis-2,6-Dimethylmorp...)
Affinity DataIC50:  12nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320534(US10174035, Compound 78 | [5-(1-Methyl-1H-pyrazol-...)
Affinity DataIC50:  13nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320473(US10174035, Compound 19 | [4-(Morpholin-4-yl)piper...)
Affinity DataIC50:  13nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320534(US10174035, Compound 78 | [5-(1-Methyl-1H-pyrazol-...)
Affinity DataIC50:  13nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320473(US10174035, Compound 19 | [4-(Morpholin-4-yl)piper...)
Affinity DataIC50:  13nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320512(US10174035, Compound 58 | [2-(1-Methyl-1H-pyrazol-...)
Affinity DataIC50:  14nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320495(US10174035, Compound 41 | [2-(1,3-Dimethyl-1H-pyra...)
Affinity DataIC50:  14nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320512(US10174035, Compound 58 | [2-(1-Methyl-1H-pyrazol-...)
Affinity DataIC50:  14nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320495(US10174035, Compound 41 | [2-(1,3-Dimethyl-1H-pyra...)
Affinity DataIC50:  14nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320569(US10174035, Compound 112 | {4-[cis-2,6-Dimethylmor...)
Affinity DataIC50:  15nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320490(N-(Cyclohexylmethyl)-2-(1-methyl-1H-pyrazol-4-yl)-...)
Affinity DataIC50:  15nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320456(US10174035, Compound 3 | [2-(1-Methyl-1H-pyrazol-4...)
Affinity DataIC50:  15nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320456(US10174035, Compound 3 | [2-(1-Methyl-1H-pyrazol-4...)
Affinity DataIC50:  15nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320572(5-(1-Methyl-1H-pyrazol-4-yl)-7-(morpholin-4-yl)-N-...)
Affinity DataIC50:  16nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320468(US10174035, Compound 14 | [4-(2-Hydroxypropan-2-yl...)
Affinity DataIC50:  16nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320468(US10174035, Compound 14 | [4-(2-Hydroxypropan-2-yl...)
Affinity DataIC50:  16nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform(Homo sapiens (Human))
Daiichi Sankyo

US Patent
LigandPNGBDBM320518(2-(1-Methyl-1H-pyrazol-4-yl)-N-{2-[1-methylpyrroli...)
Affinity DataIC50:  17nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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