Compile Data Set for Download or QSAR
maximum 50k data
Found 76 Enz. Inhib. hit(s) with all data for entry = 2229
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357915((E)-2-(((Dimethylamino)methylene)amino)-7-isopropy...)
Affinity DataIC50:  80nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357864(US10214536, Compound 24)
Affinity DataIC50:  110nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357870(US10214536, Compound 38)
Affinity DataIC50:  150nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357869(US10214536, Compound 36)
Affinity DataIC50:  160nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357894(US10214536, Compound 76)
Affinity DataIC50:  170nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357921(US10214536, Compound 288)
Affinity DataIC50:  180nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357919(US10214536, Compound 286)
Affinity DataIC50:  180nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357877(US10214536, Compound 53)
Affinity DataIC50:  190nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357872(US10214536, Compound 42)
Affinity DataIC50:  190nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357866(US10214536, Compound 28)
Affinity DataIC50:  220nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357865(US10214536, Compound 26)
Affinity DataIC50:  240nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357871(US10214536, Compound 40)
Affinity DataIC50:  240nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357896(US10214536, Compound 80)
Affinity DataIC50:  260nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357891(US10214536, Compound 69)
Affinity DataIC50:  320nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357897(US10214536, Compound 81)
Affinity DataIC50:  330nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357860(US10214536, Compound 11)
Affinity DataIC50:  340nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357889(US10214536, Compound 65)
Affinity DataIC50:  370nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357929(US10214536, Compound 296)
Affinity DataIC50:  390nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357931(US10214536, Compound 298)
Affinity DataIC50:  410nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357909(2-Amino-8-isopropyl-5-oxo-5H-chromeno[2,3-b]pyridi...)
Affinity DataIC50:  410nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357893(US10214536, Compound 74)
Affinity DataIC50:  510nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357906(Ethyl 2-amino-8-bromo-5-oxo-5H-chromeno[2,3-b]pyri...)
Affinity DataIC50:  520nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357930(US10214536, Compound 297)
Affinity DataIC50:  550nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357861(US10214536, Compound 13)
Affinity DataIC50:  560nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357859(US10214536, Compound 8)
Affinity DataIC50:  560nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357892(US10214536, Compound 71)
Affinity DataIC50:  600nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357886(2-Amino-7-(4,4-dimethylcyclohex-1-en-1-yl)-5-oxo-5...)
Affinity DataIC50:  740nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357895(US10214536, Compound 78)
Affinity DataIC50:  790nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357884(US10214536, Compound 57b)
Affinity DataIC50:  800nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357880(US10214536, Compound 55c)
Affinity DataIC50:  880nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357857(Aphthasol | US10214536, Amlexanox)
Affinity DataIC50:  980nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357901(US10214536, Compound 180)
Affinity DataIC50:  1.07E+3nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357887(US10214536, Compound 61)
Affinity DataIC50:  1.17E+3nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357874(US10214536, Compound 47)
Affinity DataIC50:  1.20E+3nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357905(2-Amino-7-isobutyl-5-oxo-5H-chromeno[2,3-b]pyridin...)
Affinity DataIC50:  1.23E+3nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357914(2-Amino-8-fluoro-7-isopropyl-5-oxo-5H-chromeno[2,3...)
Affinity DataIC50:  1.24E+3nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357927(US10214536, Compound 294)
Affinity DataIC50:  1.39E+3nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357900(US10214536, Compound 176)
Affinity DataIC50:  1.40E+3nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357922(US10214536, Compound 289)
Affinity DataIC50:  1.40E+3nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357888(Ethyl 2-amino-7-(4,4-dimethylcyclohexyl)-5-oxo-5H-...)
Affinity DataIC50:  1.41E+3nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357890(US10214536, Compound 67)
Affinity DataIC50:  1.45E+3nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357907((E)-2-Amino-8-(2-cyclopentylvinyl)-5-oxo-5H-chrome...)
Affinity DataIC50:  1.49E+3nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357858(US10214536, Compound 5)
Affinity DataIC50:  1.51E+3nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357932(US10214536, Compound 299)
Affinity DataIC50:  1.53E+3nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357898(US10214536, Compound 97)
Affinity DataIC50:  1.56E+3nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357862(US10214536, Compound 15)
Affinity DataIC50:  1.67E+3nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357904(2-Amino-7-(2-cyclobutylethyl)-5-oxo-5H-chromeno[2,...)
Affinity DataIC50:  1.67E+3nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357903(2-Amino-7-isopentyl-5-oxo-5H-chromeno[2,3-b]pyridi...)
Affinity DataIC50:  2.01E+3nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357924(US10214536, Compound 291)
Affinity DataIC50:  2.05E+3nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSerine/threonine-protein kinase TBK1(Homo sapiens (Human))
The Regents Of The University Of Michigan

US Patent
LigandPNGBDBM357912(Ethyl 2-amino-8-fluoro-5-oxo-7-(prop-1-en-2-yl)-5H...)
Affinity DataIC50:  2.16E+3nMAssay Description:Kinase assays are commonly used for determining the ability of a small molecule to inhibit enzyme activity. By measuring the degree of phosphorylatio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
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