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Found 3 Enz. Inhib. hit(s) with all data for entry = 2878
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM291282(US10280174, Compound A | US9580432, Example 13)
Affinity DataIC50:  1.19nMAssay Description:In a condition set for a method of measuring inhibitory activity in vitro of the compounds against BTK kinase activity, FL-Peptide 2 was used as a su...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM1773(US10280174, Comparative Compound 1 | US8476284, 4 ...)
Affinity DataIC50:  1.30nMAssay Description:With regard to the setting of the conditions for a method for measuring the inhibitory activity of a compound against EGFR kinase activity in vitro, ...More data for this Ligand-Target Pair
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Taiho Pharmaceutical

US Patent
LigandPNGBDBM291282(US10280174, Compound A | US9580432, Example 13)
Affinity DataIC50:  16.9nMAssay Description:With regard to the setting of the conditions for a method for measuring the inhibitory activity of a compound against EGFR kinase activity in vitro, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent