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Found 14 Enz. Inhib. hit(s) with all data for entry = 3228
TargetPotassium-transporting ATPase alpha chain 1(Sus scrofa (Pig))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM394383(N-methyl-1-[1-(phenylsulfonyl)-5-(3-thienyl)-1H-py...)
Affinity DataIC50:  4.20nMAssay Description:According to the method [Biochem. Biophys. Acta., 728, 31 (1983)] of Wallmark et al., a gastric mucous membrane microsomal fraction was prepared from...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPotassium-transporting ATPase alpha chain 1(Sus scrofa (Pig))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM394395(1-[5-(2,4-Difluorophenyl)-1-(pyridin-3-ylsulfonyl)...)
Affinity DataIC50:  8.90nMAssay Description:According to the method [Biochem. Biophys. Acta., 728, 31 (1983)] of Wallmark et al., a gastric mucous membrane microsomal fraction was prepared from...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPotassium-transporting ATPase alpha chain 1(Sus scrofa (Pig))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM394391(1-{5-(2-Fluorophenyl)-1-[(2-fluorophenyl)sulfonyl]...)
Affinity DataIC50:  9nMAssay Description:According to the method [Biochem. Biophys. Acta., 728, 31 (1983)] of Wallmark et al., a gastric mucous membrane microsomal fraction was prepared from...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPotassium-transporting ATPase alpha chain 1(Sus scrofa (Pig))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM394389(Ethyl 1-(pyridazin-3-ylsulfonyl)-5-phenyl-1H-pyrro...)
Affinity DataIC50:  13nMAssay Description:According to the method [Biochem. Biophys. Acta., 728, 31 (1983)] of Wallmark et al., a gastric mucous membrane microsomal fraction was prepared from...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPotassium-transporting ATPase alpha chain 1(Sus scrofa (Pig))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM394392(1-[5-(2-Fluorophenyl)-1-(pyridin-3-ylsulfonyl)-1H-...)
Affinity DataIC50:  22nMAssay Description:According to the method [Biochem. Biophys. Acta., 728, 31 (1983)] of Wallmark et al., a gastric mucous membrane microsomal fraction was prepared from...More data for this Ligand-Target Pair
TargetPotassium-transporting ATPase alpha chain 1(Sus scrofa (Pig))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM394388(1-[1-(1-Benzothien-2-ylsulfonyl)-5-phenyl-1H-pyrro...)
Affinity DataIC50:  33nMAssay Description:According to the method [Biochem. Biophys. Acta., 728, 31 (1983)] of Wallmark et al., a gastric mucous membrane microsomal fraction was prepared from...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPotassium-transporting ATPase alpha chain 1(Sus scrofa (Pig))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM394394(N-Methyl-1-[5-(2-methylphenyl)-1-(pyridin-3-ylsulf...)
Affinity DataIC50:  36nMAssay Description:According to the method [Biochem. Biophys. Acta., 728, 31 (1983)] of Wallmark et al., a gastric mucous membrane microsomal fraction was prepared from...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPotassium-transporting ATPase alpha chain 1(Sus scrofa (Pig))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM394386(N-Methyl-1-[5-phenyl-1-(3-thienylsulfonyl)-1H-pyrr...)
Affinity DataIC50:  51nMAssay Description:According to the method [Biochem. Biophys. Acta., 728, 31 (1983)] of Wallmark et al., a gastric mucous membrane microsomal fraction was prepared from...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPotassium-transporting ATPase alpha chain 1(Sus scrofa (Pig))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM394378(Ethyl 1-[(4-methoxyphenyl)sulfonyl]-5-phenyl-1H-py...)
Affinity DataIC50:  51nMAssay Description:According to the method [Biochem. Biophys. Acta., 728, 31 (1983)] of Wallmark et al., a gastric mucous membrane microsomal fraction was prepared from...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPotassium-transporting ATPase alpha chain 1(Sus scrofa (Pig))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM394390(1-[5-(2-Fluorophenyl)-1-{[3-(methylsulfonyl)phenyl...)
Affinity DataIC50:  62nMAssay Description:According to the method [Biochem. Biophys. Acta., 728, 31 (1983)] of Wallmark et al., a gastric mucous membrane microsomal fraction was prepared from...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPotassium-transporting ATPase alpha chain 1(Sus scrofa (Pig))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM394387(US10308605, Example 140)
Affinity DataIC50:  78nMAssay Description:According to the method [Biochem. Biophys. Acta., 728, 31 (1983)] of Wallmark et al., a gastric mucous membrane microsomal fraction was prepared from...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPotassium-transporting ATPase alpha chain 1(Sus scrofa (Pig))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM394393(N-Methyl-3-({4-[(methylamino)methyl]-2-phenyl-1H-p...)
Affinity DataIC50:  86nMAssay Description:According to the method [Biochem. Biophys. Acta., 728, 31 (1983)] of Wallmark et al., a gastric mucous membrane microsomal fraction was prepared from...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPotassium-transporting ATPase alpha chain 1(Sus scrofa (Pig))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM394377(N-Methyl-1-{5-(3-methylphenyl)-1-[(4-methylphenyl)...)
Affinity DataIC50:  91nMAssay Description:According to the method [Biochem. Biophys. Acta., 728, 31 (1983)] of Wallmark et al., a gastric mucous membrane microsomal fraction was prepared from...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPotassium-transporting ATPase alpha chain 1(Sus scrofa (Pig))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM394382(1-[(4-Methoxyphenyl)sulfonyl]-5-phenyl-1H-pyrrole-...)
Affinity DataIC50:  710nMAssay Description:According to the method [Biochem. Biophys. Acta., 728, 31 (1983)] of Wallmark et al., a gastric mucous membrane microsomal fraction was prepared from...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent