TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceutical
US Patent
Shanghai Hengrui Pharmaceutical
US Patent
Affinity DataIC50: 0.110nMAssay Description:Human: Test Example 1. Human GnRHr (GnRH Receptor) Activity Assay of the Present Compounds.In vitro GnRHr protein activity was tested by the followin...More data for this Ligand-Target Pair
TargetG_PROTEIN_RECEP_F1_2 domain-containing protein(Oryctolagus cuniculus (Rabbit))
Shanghai Hengrui Pharmaceutical
US Patent
Shanghai Hengrui Pharmaceutical
US Patent
Affinity DataIC50: 0.240nMAssay Description:Rabbit: This assay was used to determine the inhibition effect of the present compounds on the activity of rabbit GnRHr protein expressed by rabbit G...More data for this Ligand-Target Pair
TargetG_PROTEIN_RECEP_F1_2 domain-containing protein(Oryctolagus cuniculus (Rabbit))
Shanghai Hengrui Pharmaceutical
US Patent
Shanghai Hengrui Pharmaceutical
US Patent
Affinity DataIC50: 0.270nMAssay Description:Rabbit: This assay was used to determine the inhibition effect of the present compounds on the activity of rabbit GnRHr protein expressed by rabbit G...More data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceutical
US Patent
Shanghai Hengrui Pharmaceutical
US Patent
Affinity DataIC50: 0.420nMAssay Description:Human: Test Example 1. Human GnRHr (GnRH Receptor) Activity Assay of the Present Compounds.In vitro GnRHr protein activity was tested by the followin...More data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceutical
US Patent
Shanghai Hengrui Pharmaceutical
US Patent
Affinity DataIC50: 0.430nMAssay Description:Human: Test Example 1. Human GnRHr (GnRH Receptor) Activity Assay of the Present Compounds.In vitro GnRHr protein activity was tested by the followin...More data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceutical
US Patent
Shanghai Hengrui Pharmaceutical
US Patent
Affinity DataIC50: 0.490nMAssay Description:Human: Test Example 1. Human GnRHr (GnRH Receptor) Activity Assay of the Present Compounds.In vitro GnRHr protein activity was tested by the followin...More data for this Ligand-Target Pair
TargetG_PROTEIN_RECEP_F1_2 domain-containing protein(Oryctolagus cuniculus (Rabbit))
Shanghai Hengrui Pharmaceutical
US Patent
Shanghai Hengrui Pharmaceutical
US Patent
Affinity DataIC50: 0.570nMAssay Description:Rabbit: This assay was used to determine the inhibition effect of the present compounds on the activity of rabbit GnRHr protein expressed by rabbit G...More data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceutical
US Patent
Shanghai Hengrui Pharmaceutical
US Patent
Affinity DataIC50: 0.600nMAssay Description:Human: Test Example 1. Human GnRHr (GnRH Receptor) Activity Assay of the Present Compounds.In vitro GnRHr protein activity was tested by the followin...More data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceutical
US Patent
Shanghai Hengrui Pharmaceutical
US Patent
Affinity DataIC50: 0.660nMAssay Description:Human: Test Example 1. Human GnRHr (GnRH Receptor) Activity Assay of the Present Compounds.In vitro GnRHr protein activity was tested by the followin...More data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceutical
US Patent
Shanghai Hengrui Pharmaceutical
US Patent
Affinity DataIC50: 0.660nMAssay Description:Human: Test Example 1. Human GnRHr (GnRH Receptor) Activity Assay of the Present Compounds.In vitro GnRHr protein activity was tested by the followin...More data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceutical
US Patent
Shanghai Hengrui Pharmaceutical
US Patent
Affinity DataIC50: 0.900nMAssay Description:Human: Test Example 1. Human GnRHr (GnRH Receptor) Activity Assay of the Present Compounds.In vitro GnRHr protein activity was tested by the followin...More data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceutical
US Patent
Shanghai Hengrui Pharmaceutical
US Patent
Affinity DataIC50: 0.920nMAssay Description:Human: Test Example 1. Human GnRHr (GnRH Receptor) Activity Assay of the Present Compounds.In vitro GnRHr protein activity was tested by the followin...More data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceutical
US Patent
Shanghai Hengrui Pharmaceutical
US Patent
Affinity DataIC50: 0.960nMAssay Description:Human: Test Example 1. Human GnRHr (GnRH Receptor) Activity Assay of the Present Compounds.In vitro GnRHr protein activity was tested by the followin...More data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceutical
US Patent
Shanghai Hengrui Pharmaceutical
US Patent
Affinity DataIC50: 1.46nMAssay Description:Human: Test Example 1. Human GnRHr (GnRH Receptor) Activity Assay of the Present Compounds.In vitro GnRHr protein activity was tested by the followin...More data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceutical
US Patent
Shanghai Hengrui Pharmaceutical
US Patent
Affinity DataIC50: 2.24nMAssay Description:Human: Test Example 1. Human GnRHr (GnRH Receptor) Activity Assay of the Present Compounds.In vitro GnRHr protein activity was tested by the followin...More data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceutical
US Patent
Shanghai Hengrui Pharmaceutical
US Patent
Affinity DataIC50: 2.32nMAssay Description:Human: Test Example 1. Human GnRHr (GnRH Receptor) Activity Assay of the Present Compounds.In vitro GnRHr protein activity was tested by the followin...More data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Shanghai Hengrui Pharmaceutical
US Patent
Shanghai Hengrui Pharmaceutical
US Patent
Affinity DataIC50: 4.95nMAssay Description:Human: Test Example 1. Human GnRHr (GnRH Receptor) Activity Assay of the Present Compounds.In vitro GnRHr protein activity was tested by the followin...More data for this Ligand-Target Pair
TargetGonadotropin releasing hormone receptor(Macaca fascicularis (Crab-eating macaque) (Cynomol...)
Shanghai Hengrui Pharmaceutical
US Patent
Shanghai Hengrui Pharmaceutical
US Patent
Affinity DataIC50: 23.2nMAssay Description:Monkey: This assay was used to determine the inhibition effect of the present compounds on the activity of monkey GnRHr protein expressed by monkey G...More data for this Ligand-Target Pair
TargetGonadotropin releasing hormone receptor(Macaca fascicularis (Crab-eating macaque) (Cynomol...)
Shanghai Hengrui Pharmaceutical
US Patent
Shanghai Hengrui Pharmaceutical
US Patent
Affinity DataIC50: 78.6nMAssay Description:Monkey: This assay was used to determine the inhibition effect of the present compounds on the activity of monkey GnRHr protein expressed by monkey G...More data for this Ligand-Target Pair