Compile Data Set for Download or QSAR
maximum 50k data
Found 12 Enz. Inhib. hit(s) with all data for entry = 8854
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
The Industry & Academic Cooperation In Chungnam National University (IAC)

US Patent
LigandPNGBDBM423394(US10501473, Example 36)
Affinity DataIC50:  17.7nMAssay Description:RIPK1 protein was over-expressed in HEK293 cell line, to which lysis buffer (50 mM Tris-Cl [pH 8.0], 150 mM NaCl, 1 mM EDTA, 1% NP-40, 0.4 mM phenylm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
The Industry & Academic Cooperation In Chungnam National University (IAC)

US Patent
LigandPNGBDBM423407(US10501473, Example 76)
Affinity DataIC50:  61.2nMAssay Description:RIPK1 protein was over-expressed in HEK293 cell line, to which lysis buffer (50 mM Tris-Cl [pH 8.0], 150 mM NaCl, 1 mM EDTA, 1% NP-40, 0.4 mM phenylm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
The Industry & Academic Cooperation In Chungnam National University (IAC)

US Patent
LigandPNGBDBM423404(US10501473, Example 74)
Affinity DataIC50:  65.6nMAssay Description:RIPK1 protein was over-expressed in HEK293 cell line, to which lysis buffer (50 mM Tris-Cl [pH 8.0], 150 mM NaCl, 1 mM EDTA, 1% NP-40, 0.4 mM phenylm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
The Industry & Academic Cooperation In Chungnam National University (IAC)

US Patent
LigandPNGBDBM423405(US10501473, Example 75)
Affinity DataIC50:  73.4nMAssay Description:RIPK1 protein was over-expressed in HEK293 cell line, to which lysis buffer (50 mM Tris-Cl [pH 8.0], 150 mM NaCl, 1 mM EDTA, 1% NP-40, 0.4 mM phenylm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
The Industry & Academic Cooperation In Chungnam National University (IAC)

US Patent
LigandPNGBDBM36371(5-(1H-indol-3-ylmethyl)-3-methyl-2-thioxo-4-Imidaz...)
Affinity DataIC50:  95.5nMAssay Description:RIPK1 protein was over-expressed in HEK293 cell line, to which lysis buffer (50 mM Tris-Cl [pH 8.0], 150 mM NaCl, 1 mM EDTA, 1% NP-40, 0.4 mM phenylm...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
The Industry & Academic Cooperation In Chungnam National University (IAC)

US Patent
LigandPNGBDBM423379(US10501473, Example 30)
Affinity DataIC50:  102nMAssay Description:RIPK1 protein was over-expressed in HEK293 cell line, to which lysis buffer (50 mM Tris-Cl [pH 8.0], 150 mM NaCl, 1 mM EDTA, 1% NP-40, 0.4 mM phenylm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
The Industry & Academic Cooperation In Chungnam National University (IAC)

US Patent
LigandPNGBDBM423400(US10501473, Example 39)
Affinity DataIC50:  193nMAssay Description:RIPK1 protein was over-expressed in HEK293 cell line, to which lysis buffer (50 mM Tris-Cl [pH 8.0], 150 mM NaCl, 1 mM EDTA, 1% NP-40, 0.4 mM phenylm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
The Industry & Academic Cooperation In Chungnam National University (IAC)

US Patent
LigandPNGBDBM423401(US10501473, Example 51)
Affinity DataIC50:  217nMAssay Description:RIPK1 protein was over-expressed in HEK293 cell line, to which lysis buffer (50 mM Tris-Cl [pH 8.0], 150 mM NaCl, 1 mM EDTA, 1% NP-40, 0.4 mM phenylm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
The Industry & Academic Cooperation In Chungnam National University (IAC)

US Patent
LigandPNGBDBM423403(US10501473, Example 63)
Affinity DataIC50:  230nMAssay Description:RIPK1 protein was over-expressed in HEK293 cell line, to which lysis buffer (50 mM Tris-Cl [pH 8.0], 150 mM NaCl, 1 mM EDTA, 1% NP-40, 0.4 mM phenylm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
The Industry & Academic Cooperation In Chungnam National University (IAC)

US Patent
LigandPNGBDBM423389(US10501473, Example 35)
Affinity DataIC50:  360nMAssay Description:RIPK1 protein was over-expressed in HEK293 cell line, to which lysis buffer (50 mM Tris-Cl [pH 8.0], 150 mM NaCl, 1 mM EDTA, 1% NP-40, 0.4 mM phenylm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
The Industry & Academic Cooperation In Chungnam National University (IAC)

US Patent
LigandPNGBDBM423376(US10501473, Example 4)
Affinity DataIC50:  1.13E+3nMAssay Description:RIPK1 protein was over-expressed in HEK293 cell line, to which lysis buffer (50 mM Tris-Cl [pH 8.0], 150 mM NaCl, 1 mM EDTA, 1% NP-40, 0.4 mM phenylm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetReceptor-interacting serine/threonine-protein kinase 1(Homo sapiens (Human))
The Industry & Academic Cooperation In Chungnam National University (IAC)

US Patent
LigandPNGBDBM423402(US10501473, Example 52)
Affinity DataIC50:  8.17E+3nMAssay Description:RIPK1 protein was over-expressed in HEK293 cell line, to which lysis buffer (50 mM Tris-Cl [pH 8.0], 150 mM NaCl, 1 mM EDTA, 1% NP-40, 0.4 mM phenylm...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent