Compile Data Set for Download or QSAR
maximum 50k data
Found 9 Enz. Inhib. hit(s) with all data for entry = 9069
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Eli Lilly

US Patent
LigandPNGBDBM438836(1'-[1-(4- Cyanophenyl)ethyl]- 5,5- spirocyclopropa...)
Affinity DataKi:  6nMAssay Description:His-tagged human RAR-related orphan receptor alpha (hRORa), human RAR-related orphan receptor beta (hRORb), and human RAR-related orphan receptor gam...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Eli Lilly

US Patent
LigandPNGBDBM438835(N-{[5-(Ethylsulfonyl)pyridin-2-yl]methyl}-1″...)
Affinity DataKi:  6.40nMAssay Description:His-tagged human RAR-related orphan receptor alpha (hRORa), human RAR-related orphan receptor beta (hRORb), and human RAR-related orphan receptor gam...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Eli Lilly

US Patent
LigandPNGBDBM438834(N-{[5-(Ethylsulfonyl)pyridin-2-yl]methyl}-5′...)
Affinity DataKi:  6.96nMAssay Description:His-tagged human RAR-related orphan receptor alpha (hRORa), human RAR-related orphan receptor beta (hRORb), and human RAR-related orphan receptor gam...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-alpha(Homo sapiens (Human))
Eli Lilly

US Patent
LigandPNGBDBM438835(N-{[5-(Ethylsulfonyl)pyridin-2-yl]methyl}-1″...)
Affinity DataKi:  3.46E+3nMAssay Description:His-tagged human RAR-related orphan receptor alpha (hRORa), human RAR-related orphan receptor beta (hRORb), and human RAR-related orphan receptor gam...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-alpha(Homo sapiens (Human))
Eli Lilly

US Patent
LigandPNGBDBM438834(N-{[5-(Ethylsulfonyl)pyridin-2-yl]methyl}-5′...)
Affinity DataKi:  5.68E+3nMAssay Description:His-tagged human RAR-related orphan receptor alpha (hRORa), human RAR-related orphan receptor beta (hRORb), and human RAR-related orphan receptor gam...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRAR related orphan receptor B isoform 1(Human)
Eli Lilly

US Patent
LigandPNGBDBM438834(N-{[5-(Ethylsulfonyl)pyridin-2-yl]methyl}-5′...)
Affinity DataKi: >1.25E+4nMAssay Description:His-tagged human RAR-related orphan receptor alpha (hRORa), human RAR-related orphan receptor beta (hRORb), and human RAR-related orphan receptor gam...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRAR related orphan receptor B isoform 1(Human)
Eli Lilly

US Patent
LigandPNGBDBM438835(N-{[5-(Ethylsulfonyl)pyridin-2-yl]methyl}-1″...)
Affinity DataKi: >1.25E+4nMAssay Description:His-tagged human RAR-related orphan receptor alpha (hRORa), human RAR-related orphan receptor beta (hRORb), and human RAR-related orphan receptor gam...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRAR related orphan receptor B isoform 1(Human)
Eli Lilly

US Patent
LigandPNGBDBM438836(1'-[1-(4- Cyanophenyl)ethyl]- 5,5- spirocyclopropa...)
Affinity DataKi: >1.25E+4nMAssay Description:His-tagged human RAR-related orphan receptor alpha (hRORa), human RAR-related orphan receptor beta (hRORb), and human RAR-related orphan receptor gam...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-alpha(Homo sapiens (Human))
Eli Lilly

US Patent
LigandPNGBDBM438836(1'-[1-(4- Cyanophenyl)ethyl]- 5,5- spirocyclopropa...)
Affinity DataKi: >2.04E+4nMAssay Description:His-tagged human RAR-related orphan receptor alpha (hRORa), human RAR-related orphan receptor beta (hRORb), and human RAR-related orphan receptor gam...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent