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Found 22 Enz. Inhib. hit(s) with all data for entry = 9820
TargetProgrammed cell death 1 ligand/protein 1(Homo sapiens)
Institute Of Materia Medica, Chinese Academy Of Medical Sciences

US Patent
LigandPNGBDBM491037((S)—N-(4-(2-bromo-3-phenylbenzyloxy)-5-chloro-2-(p...)
Affinity DataIC50: <0.000100nMAssay Description:In vitro activity evaluation: Cisbio PD-1/PD-L1 binding assay kit was applied for the detection method of in vitro enzymology level.Screening Princip...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetProgrammed cell death protein 1(Homo sapiens)
Institute Of Materia Medica, Chinese Academy Of Medical Sciences

US Patent
LigandPNGBDBM491057(N-(4-(2-bromo-3-phenylbenzyloxy)-5-chloro-2-(pyrid...)
Affinity DataIC50:  0.000500nMAssay Description:In vitro activity evaluation: Cisbio PD-1/PD-L1 binding assay kit was applied for the detection method of in vitro enzymology level.Screening Princip...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetProgrammed cell death 1 ligand/protein 1(Homo sapiens)
Institute Of Materia Medica, Chinese Academy Of Medical Sciences

US Patent
LigandPNGBDBM491049((E)-3-(4-(2-bromo-3-phenylbenzyloxy)-5-chloro-2-(p...)
Affinity DataIC50:  2.33nMAssay Description:In vitro activity evaluation: Cisbio PD-1/PD-L1 binding assay kit was applied for the detection method of in vitro enzymology level.Screening Princip...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetProgrammed cell death 1 ligand/protein 1(Homo sapiens)
Institute Of Materia Medica, Chinese Academy Of Medical Sciences

US Patent
LigandPNGBDBM491056(N-(4-(2-bromo-3-phenylbenzyloxy)-5-chloro-2-(pyrid...)
Affinity DataIC50:  5.29nMAssay Description:In vitro activity evaluation: Cisbio PD-1/PD-L1 binding assay kit was applied for the detection method of in vitro enzymology level.Screening Princip...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetProgrammed cell death 1 ligand/protein 1(Homo sapiens)
Institute Of Materia Medica, Chinese Academy Of Medical Sciences

US Patent
LigandPNGBDBM491040((S)—N-(4-(2-chloro-3-phenylbenzyloxy)-5-chloro-2-(...)
Affinity DataIC50:  40.1nMAssay Description:In vitro activity evaluation: Cisbio PD-1/PD-L1 binding assay kit was applied for the detection method of in vitro enzymology level.Screening Princip...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetProgrammed cell death 1 ligand/protein 1(Homo sapiens)
Institute Of Materia Medica, Chinese Academy Of Medical Sciences

US Patent
LigandPNGBDBM491043(N-(4-(2-bromo-3-phenylbenzyloxy)-5-chloro-2-(pyrid...)
Affinity DataIC50:  41.1nMAssay Description:In vitro activity evaluation: Cisbio PD-1/PD-L1 binding assay kit was applied for the detection method of in vitro enzymology level.Screening Princip...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetProgrammed cell death 1 ligand/protein 1(Homo sapiens)
Institute Of Materia Medica, Chinese Academy Of Medical Sciences

US Patent
LigandPNGBDBM491039((R)—N-(4-(2-bromo-3-phenylbenzyloxy)-5-chloro-2-(p...)
Affinity DataIC50:  42.9nMAssay Description:In vitro activity evaluation: Cisbio PD-1/PD-L1 binding assay kit was applied for the detection method of in vitro enzymology level.Screening Princip...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetProgrammed cell death 1 ligand/protein 1(Homo sapiens)
Institute Of Materia Medica, Chinese Academy Of Medical Sciences

US Patent
LigandPNGBDBM491046(N,N-bis(2-hydroxyethyl)-4-(2-bromo-3-phenylbenzylo...)
Affinity DataIC50:  51nMAssay Description:In vitro activity evaluation: Cisbio PD-1/PD-L1 binding assay kit was applied for the detection method of in vitro enzymology level.Screening Princip...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetProgrammed cell death 1 ligand/protein 1(Homo sapiens)
Institute Of Materia Medica, Chinese Academy Of Medical Sciences

US Patent
LigandPNGBDBM491055(N-(hydroxyethyl)-4-(2-bromo-3-phenylbenzyloxy)-5-c...)
Affinity DataIC50:  53.8nMAssay Description:In vitro activity evaluation: Cisbio PD-1/PD-L1 binding assay kit was applied for the detection method of in vitro enzymology level.Screening Princip...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetProgrammed cell death 1 ligand/protein 1(Homo sapiens)
Institute Of Materia Medica, Chinese Academy Of Medical Sciences

US Patent
LigandPNGBDBM491051(N-(4-(2-bromo-3-phenylbenzyloxy)-5-chloro-2-(pyrid...)
Affinity DataIC50:  61nMAssay Description:In vitro activity evaluation: Cisbio PD-1/PD-L1 binding assay kit was applied for the detection method of in vitro enzymology level.Screening Princip...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetProgrammed cell death 1 ligand/protein 1(Homo sapiens)
Institute Of Materia Medica, Chinese Academy Of Medical Sciences

US Patent
LigandPNGBDBM491038((S)-isopropyl N-(4-(2-bromo-3-phenylbenzyloxy)-5-c...)
Affinity DataIC50:  82.3nMAssay Description:In vitro activity evaluation: Cisbio PD-1/PD-L1 binding assay kit was applied for the detection method of in vitro enzymology level.Screening Princip...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetProgrammed cell death 1 ligand/protein 1(Homo sapiens)
Institute Of Materia Medica, Chinese Academy Of Medical Sciences

US Patent
LigandPNGBDBM491041((S)—N-(4-(2-fluoro-3-phenylbenzyloxy)-5-chloro-2-(...)
Affinity DataIC50:  134nMAssay Description:In vitro activity evaluation: Cisbio PD-1/PD-L1 binding assay kit was applied for the detection method of in vitro enzymology level.Screening Princip...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetProgrammed cell death 1 ligand/protein 1(Homo sapiens)
Institute Of Materia Medica, Chinese Academy Of Medical Sciences

US Patent
LigandPNGBDBM491036(Ethyl N-(4-(2-bromo-3-phenylbenzyloxy)-5-chloro-2-...)
Affinity DataIC50:  148nMAssay Description:In vitro activity evaluation: Cisbio PD-1/PD-L1 binding assay kit was applied for the detection method of in vitro enzymology level.Screening Princip...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetProgrammed cell death 1 ligand/protein 1(Homo sapiens)
Institute Of Materia Medica, Chinese Academy Of Medical Sciences

US Patent
LigandPNGBDBM491047(N-(2-methanesulfonaminoethyl)-4-(2-bromo-3-phenylb...)
Affinity DataIC50:  199nMAssay Description:In vitro activity evaluation: Cisbio PD-1/PD-L1 binding assay kit was applied for the detection method of in vitro enzymology level.Screening Princip...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetProgrammed cell death 1 ligand/protein 1(Homo sapiens)
Institute Of Materia Medica, Chinese Academy Of Medical Sciences

US Patent
LigandPNGBDBM491044(N-(4-(2-bromo-3-phenylbenzyloxy)-5-chloro-2-(pyrid...)
Affinity DataIC50:  200nMAssay Description:In vitro activity evaluation: Cisbio PD-1/PD-L1 binding assay kit was applied for the detection method of in vitro enzymology level.Screening Princip...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProgrammed cell death 1 ligand/protein 1(Homo sapiens)
Institute Of Materia Medica, Chinese Academy Of Medical Sciences

US Patent
LigandPNGBDBM491042((S)—N-(4-(3-phenylbenzyloxy)-5-chloro-2-(pyridin-3...)
Affinity DataIC50:  318nMAssay Description:In vitro activity evaluation: Cisbio PD-1/PD-L1 binding assay kit was applied for the detection method of in vitro enzymology level.Screening Princip...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProgrammed cell death 1 ligand/protein 1(Homo sapiens)
Institute Of Materia Medica, Chinese Academy Of Medical Sciences

US Patent
LigandPNGBDBM491052(N-(4-(2-bromo-3-phenylbenzyloxy)-5-chloro-2-(pyrid...)
Affinity DataIC50:  406nMAssay Description:In vitro activity evaluation: Cisbio PD-1/PD-L1 binding assay kit was applied for the detection method of in vitro enzymology level.Screening Princip...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetProgrammed cell death 1 ligand/protein 1(Homo sapiens)
Institute Of Materia Medica, Chinese Academy Of Medical Sciences

US Patent
LigandPNGBDBM491048(N-(2-acetylaminoethyl)-4-(2-bromo-3-phenylbenzylox...)
Affinity DataIC50:  551nMAssay Description:In vitro activity evaluation: Cisbio PD-1/PD-L1 binding assay kit was applied for the detection method of in vitro enzymology level.Screening Princip...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProgrammed cell death 1 ligand/protein 1(Homo sapiens)
Institute Of Materia Medica, Chinese Academy Of Medical Sciences

US Patent
LigandPNGBDBM491054(N-(4-(2-bromo-3-phenylbenzyloxy)-5-chloro-2-(pyrid...)
Affinity DataIC50:  835nMAssay Description:In vitro activity evaluation: Cisbio PD-1/PD-L1 binding assay kit was applied for the detection method of in vitro enzymology level.Screening Princip...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProgrammed cell death 1 ligand/protein 1(Homo sapiens)
Institute Of Materia Medica, Chinese Academy Of Medical Sciences

US Patent
LigandPNGBDBM491053(N-(4-(2-bromo-3-phenylbenzyloxy)-5-chloro-2-(pyrid...)
Affinity DataIC50:  4.99E+3nMAssay Description:In vitro activity evaluation: Cisbio PD-1/PD-L1 binding assay kit was applied for the detection method of in vitro enzymology level.Screening Princip...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetProgrammed cell death 1 ligand/protein 1(Homo sapiens)
Institute Of Materia Medica, Chinese Academy Of Medical Sciences

US Patent
LigandPNGBDBM491050(2-(4-(2-bromo-3-phenylbenzyloxy)-5-chloro-2-(pyrid...)
Affinity DataIC50:  1.62E+4nMAssay Description:In vitro activity evaluation: Cisbio PD-1/PD-L1 binding assay kit was applied for the detection method of in vitro enzymology level.Screening Princip...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
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TargetProgrammed cell death 1 ligand/protein 1(Homo sapiens)
Institute Of Materia Medica, Chinese Academy Of Medical Sciences

US Patent
LigandPNGBDBM491045((E)-3-(4-(2-bromo-3-phenylbenzyloxy)-5-chloro-2-(p...)
Affinity DataIC50:  2.69E+4nMAssay Description:In vitro activity evaluation: Cisbio PD-1/PD-L1 binding assay kit was applied for the detection method of in vitro enzymology level.Screening Princip...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent