Compile Data Set for Download or QSAR
maximum 50k data
Found 178 Enz. Inhib. hit(s) with all data for entry = 9894
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497228((1S,4R)-4-(5-(1-((1- methylpiperidin-4- yl)sulfony...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497229((1S,4R)-4-(2-(((S)-pentan- 2-yl)amino)-5-(1- ((tet...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497230((1S,4R)-4-(2-(((S)-pentan- 2-yl)amino)-5-(1- (pipe...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497231((1S,4R)-4-(5-(1-((2- methoxyethyl)sulfonyl) piperi...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497232((1S,4R)-4-(5-(1- (methylsulfonyl)piperidin- 4-yl)-...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497233((4-(7-((1R,4S)-4- hydroxycyclohexyl)-2- (((S)-pent...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497236(1-(4-(7-((1R,4S)-4- hydroxycyclohexyl)-2- (((S)-pe...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497237((4-(7-((1R,4S)-4- hydroxycyclohexyl)-2- (((S)-pent...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497238((4-(7-((1R,4S)-4- hydroxycyclohexyl)-2- (((S)-pent...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497241(Azetidin-3-yl(4-(7- ((1R,4S)-4- hydroxycyclohexyl)...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497242((4-(7-((1R,4S)-4- hydroxycyclohexyl)-2- (((S)-pent...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497243(7-((1R,4S)-4- hydroxycyclohexyl)-2- (((S)-pentan-2...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497244(7-((1R,4S)-4- hydroxycyclohexyl)-5-(1- (methylprol...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497245((4-(7-((1R,4S)-4- hydroxycyclohexyl)-2- (((S)-pent...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497246((4-(7-((1R,4S)-4- hydroxycyclohexyl)-2- (((S)-pent...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497247((4-(7-((1R,4S)-4- hydroxycyclohexyl)-2- (((S)-pent...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497247((4-(7-((1R,4S)-4- hydroxycyclohexyl)-2- (((S)-pent...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497250((4-(7-((1R,4S)-4- hydroxycyclohexyl)-2- (((S)-pent...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497253((4-(7-((1R,4S)-4- hydroxycyclohexyl)-2- (((S)-pent...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497254((4-(7-((1R,4S)-4- hydroxycyclohexyl)-2- (((S)-pent...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497255((4-(7-((1R,4S)-4- hydroxycyclohexyl)-2- (((S)-pent...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497258((4-(7-((1r,4S)-4- hydroxycyclohexyl)-2- (((S)-pent...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497259((4-(7-((1R,4S)-4- hydroxycyclohexyl)-2- (((S)-pent...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497260((4-(7-((1R,4S)-4- hydroxycyclohexyl)-2- (((S)-pent...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497261((4-(7-((1R,4S)-4- hydroxycyclohexyl)-2- (((S)-pent...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497262((4-(7-((1R,4S)-4- hydroxycyclohexyl)-2- (((S)-pent...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497263((4-(7-((1R,4S)-4- hydroxycyclohexyl)-2- (((S)-pent...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497264((4-(7-((1R,4S)-4- hydroxycyclohexyl)-2- (((S)-pent...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497265((4-(7-((1R,4S)-4- hydroxycyclohexyl)-2- (((S)-pent...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497266((4-(7-((1R,4S)-4- hydroxycyclohexyl)-2- (((S)-pent...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497267((2,6-dimethylpyridin-4- yl)(4-(7-((1R,4S)-4- hydro...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497268((4-(7-((1R,4S)-4- hydroxycyclohexyl)-2- (((S)-pent...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497269((1-(2-fluoroethyl)piperidin- 4-yl)(4-(7-((1R,4S)-4...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497270((4-(2-(((1S,2S)-2- ethylcyclopropyl)amino)-7- ((1R...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497271((4-(2-(((1R,2R)-2- ethylcyclopropyl)amino)-7- ((1R...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497272((1S,4R)-4-(5-([1,4'- bipiperidin]-4-yl)-2-(((S)- p...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497273((1S,4R)-4-(5-(1'-methyl- [1,4'-bipiperidin]-4-yl)-...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497274((1S,4R)-4-(2-(((S)-pentan- 2-yl)amino)-5-(1- (pipe...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497275((1S,4R)-4-(5-(1-((1- methylpiperidin-4- yl)methyl)...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497276((2,6-dimethylpyridin-4- yl)(4-(2-(((1S,2S)-2- ethy...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497277((2,6-dimethylpyridin-4- yl)(4-(2-(((1R,2R)-2- ethy...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497278((4-(7-((1r,4S)-4- hydroxycyclohexyl)-2- (((S)-pent...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497279((4-(7-((1r,4S)-4- hydroxycyclohexyl)-2- (((S)-pent...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497280((4-(7-((1r,4S)-4- hydroxycyclohexyl)-2- (((S)-pent...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497281((4-(7-((1r,4S)-4- hydroxycyclohexyl)-2- (((S)-pent...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497282((4-(7-((1r,4S)-4- hydroxycyclohexyl)-2- (((S)-pent...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497283((4-(7-((1r,4S)-4- hydroxycyclohexyl)-2- (((S)-pent...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497284((4-(7-((1r,4S)-4- hydroxycyclohexyl)-2- (((S)-pent...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497285((4-(7-((1r,4S)-4- hydroxycyclohexyl)-2- (((S)-pent...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTyrosine-protein kinase Mer(Homo sapiens (Human))
The University Of North Carolina At Chapel Hill

US Patent
LigandPNGBDBM497286((4-(7-((1r,4S)-4- hydroxycyclohexyl)-2- (((S)-pent...)
Affinity DataIC50: <3nMAssay Description:Activity Against Mer Tyrosine Kinase.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Displayed 1 to 50 (of 178 total ) | Next | Last >>
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