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Found 34 Enz. Inhib. hit(s) with all data for entry = 5906
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM99936(US8501729, 32)
Affinity DataKi:  1nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM99930(US8501729, 25)
Affinity DataKi:  1nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM99926(US8501729, 21)
Affinity DataKi:  1nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM50334453((S)-5-methyl-2-(quinuclidin-3-yl)-2,3-dihydropyrro...)
Affinity DataKi:  1nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM99935(US8501729, 31)
Affinity DataKi:  1nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM50334445((S)-2-ethyl-7-(quinuclidin-3-yl)-7,8-dihydropyrazo...)
Affinity DataKi:  1nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM50334442((S)-2-methyl-7-(quinuclidin-3-yl)-7,8-dihydropyraz...)
Affinity DataKi:  1nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM50334439((R)-2-methyl-7-(quinuclidin-3-yl)-7,8-dihydropyraz...)
Affinity DataKi:  2nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM99931(US8501729, 26)
Affinity DataKi:  2nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM50334447((S)-2-isopropyl-7-(quinuclidin-3-yl)-7,8-dihydropy...)
Affinity DataKi:  2nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM99929(US8501729, 24)
Affinity DataKi:  2nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM50334448((S)-2-isobutyl-7-(quinuclidin-3-yl)-7,8-dihydropyr...)
Affinity DataKi:  2nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM50334444((R)-2-ethyl-7-(quinuclidin-3-yl)-7,8-dihydropyrazo...)
Affinity DataKi:  2nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM50334443((R)-4-fluoro-2-methyl-7-(quinuclidin-3-yl)-7,8-dih...)
Affinity DataKi:  2nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM99932(US8501729, 27)
Affinity DataKi:  2nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM99934(US8501729, 29)
Affinity DataKi:  3nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM50334446((R)-2-isopropyl-7-(quinuclidin-3-yl)-7,8-dihydropy...)
Affinity DataKi:  3nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM99928(US8501729, 23)
Affinity DataKi:  4nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM50334449((R)-2-benzyl-7-(quinuclidin-3-yl)-7,8-dihydropyraz...)
Affinity DataKi:  5nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM50334440((R)-7-(quinuclidin-3-yl)-7,8-dihydropyrazolo[3,4,5...)
Affinity DataKi:  5nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM50334441((S)-7-(quinuclidin-3-yl)-7,8-dihydropyrazolo[3,4,5...)
Affinity DataKi:  5nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM50334451((S)-2-(4-fluorophenyl)-7-(quinuclidin-3-yl)-7,8-di...)
Affinity DataKi:  7nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM99938(US8501729, 34)
Affinity DataKi:  8nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM99939(US8501729, 35)
Affinity DataKi:  13nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM99923(US8501729, 5)
Affinity DataKi:  13nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM99942(US8501729, 30)
Affinity DataKi:  25nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM50334450((R)-2-(4-fluorophenyl)-7-(quinuclidin-3-yl)-7,8-di...)
Affinity DataKi:  29nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM99927(US8501729, 22)
Affinity DataKi:  34nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM99937(US8501729, 33)
Affinity DataKi:  49nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM99925(US8501729, 20)
Affinity DataKi:  57nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM99941(US8501729, 38)
Affinity DataKi:  59nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM99924(US8501729, 19)
Affinity DataKi:  68nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM99933(US8501729, 28)
Affinity DataKi:  108nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 3A(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM99940(US8501729, 37)
Affinity DataKi:  267nMpH: 7.5Assay Description:The relative affinity of the various compounds for the human 5-HT3 receptor was measured in a radioligand binding assay, using a scintillation proxim...More data for this Ligand-Target Pair
In DepthDetails US Patent