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Found 97 Enz. Inhib. hit(s) with all data for entry = 5966
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM50308460((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(thiophen-3-yl)...)
Affinity DataIC50:  3.51nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM50308448(2-(2-Chloro-5-((2S,3S,4R,5R,6R)-3,4,5-tris(benzylo...)
Affinity DataIC50:  4.06nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM103019(US8541380, 97)
Affinity DataIC50:  5.55nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM50308450((2S,3R,4R,5S,6R)-2-(4-chloro-3-((5-(furan-2-yl)-1,...)
Affinity DataIC50:  7.03nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM50308454((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(5-phenylfuran-...)
Affinity DataIC50:  10.6nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM103015(US8541380, 93)
Affinity DataIC50:  10.7nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM50308436((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(methylthio)-1,...)
Affinity DataIC50:  10.9nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM50319070((2S,3R,4R,5S,6R)-2-(3-((6-(1,3,4-thiadiazol-2-yl)p...)
Affinity DataIC50:  11.4nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM50319048((2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-(methylthio)pyr...)
Affinity DataIC50:  13.4nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM50308459((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(thiophen-2-yl)...)
Affinity DataIC50:  14.4nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM50308440((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-phenyl-1,3,4-th...)
Affinity DataIC50:  16.6nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM50319044((2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-(pentyloxy)pyri...)
Affinity DataIC50:  17nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM50319045((2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-(hexyloxy)pyrid...)
Affinity DataIC50:  17.3nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM103018(US8541380, 96)
Affinity DataIC50:  17.6nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM50308451((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(furan-3-yl)-1,...)
Affinity DataIC50:  17.7nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM50308463((2S,3R,4R,5S,6R)-2-(4-chloro-3-((5-(5-chlorothioph...)
Affinity DataIC50:  18.2nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM50308465((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(thiazol-4-yl)-...)
Affinity DataIC50:  21.8nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM103016(US8541380, 94)
Affinity DataIC50:  24.8nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM103013(US8541380, 91)
Affinity DataIC50:  24.9nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM102998(US8541380, 23)
Affinity DataIC50:  24.9nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM50308442((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(pyridin-2-yl)-...)
Affinity DataIC50:  30.3nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM50308445((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(2-methylpyridi...)
Affinity DataIC50:  36.4nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM50319039((2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-ethoxypyridazin...)
Affinity DataIC50:  43nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM50308464((2S,3R,4R,5S,6R)-2-(3-((5-(Benzo[b]thiophen-2-yl)-...)
Affinity DataIC50:  44.5nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM102996(US8541380, 21)
Affinity DataIC50:  45.3nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM103006(US8541380, 56)
Affinity DataIC50:  50.5nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM102995(US8541380, 20)
Affinity DataIC50:  53nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM50308453((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(5-methylfuran-...)
Affinity DataIC50:  58.3nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM50319060((2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-(furan-3-yl)pyr...)
Affinity DataIC50:  61.3nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM50319059((2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-(furan-2-yl)pyr...)
Affinity DataIC50:  64.3nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM50319067((2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-(pyridin-3-yl)p...)
Affinity DataIC50:  64.9nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM50319040((2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-propoxypyridazi...)
Affinity DataIC50:  70.8nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM50319049((2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-(ethylthio)pyri...)
Affinity DataIC50:  71.3nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM50319061((2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-(thiophen-2-yl)...)
Affinity DataIC50:  71.4nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM102994(US8541380, 14)
Affinity DataIC50:  72.6nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM50319062((2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-(thiophen-3-yl)...)
Affinity DataIC50:  75.4nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM50319047((2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-(tetrahydro-2H-...)
Affinity DataIC50:  77.6nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM50308446((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(isoquinolin-3-...)
Affinity DataIC50:  81.6nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM50319068((2S,3R,4R,5S,6R)-2-(3-((6-(benzo[d][1,3]dioxol-5-y...)
Affinity DataIC50:  82.7nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM103014(US8541380, 92)
Affinity DataIC50:  88.9nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM50308444((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(6-methylpyridi...)
Affinity DataIC50:  97.4nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM50319069((2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-(2,3-dihydroben...)
Affinity DataIC50:  103nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM102997(US8541380, 22)
Affinity DataIC50:  103nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM50308452((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(3-methylfuran-...)
Affinity DataIC50:  106nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM50319042((2S,3R,4R,5S,6R)-2-(3-((6-butoxypyridazin-3-yl)met...)
Affinity DataIC50:  109nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM50319041((2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-isopropoxypyrid...)
Affinity DataIC50:  110nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM50319046((2S,3R,4R,5S,6R)-2-(4-chloro-3-((6-(cyclohexyloxy)...)
Affinity DataIC50:  111nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM50308457(((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(1-methyl-1Hpy...)
Affinity DataIC50:  119nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM50308484((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-heptyl-1,3,4-th...)
Affinity DataIC50:  122nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetSodium/glucose cotransporter 2(Homo sapiens (Human))
Green Cross

US Patent
LigandPNGBDBM50308441((2S,3R,4R,5S,6R)-2-(4-Chloro-3-((5-(4-chlorophenyl...)
Affinity DataIC50:  126nMAssay Description:Inhibition assay using hSGLT2.More data for this Ligand-Target Pair
In DepthDetails US Patent
Displayed 1 to 50 (of 97 total ) | Next | Last >>
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