Compile Data Set for Download or QSAR
maximum 50k data
Found 7 Enz. Inhib. hit(s) with all data for entry = 6003
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM103943(US8569318, 1.1(1))
Affinity DataKi:  2.14nM IC50:  46.1nMAssay Description:Activity test of serotonin 5-HT6 receptor antagonists of the general formulas 1, 2 in the setting of competitive binding to serotonin 5-HT6 receptors...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM103944(US8569318, 1.2(2))
Affinity DataKi:  7.70nM IC50:  16.6nMAssay Description:Activity test of serotonin 5-HT6 receptor antagonists of the general formulas 1, 2 in the setting of competitive binding to serotonin 5-HT6 receptors...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM103945(US8569318, 1.2(6))
Affinity DataKi:  11.1nM IC50:  23.9nMAssay Description:Activity test of serotonin 5-HT6 receptor antagonists of the general formulas 1, 2 in the setting of competitive binding to serotonin 5-HT6 receptors...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM50396228(CHEMBL2172183 | US8569318, 1.2(3))
Affinity DataKi:  35.7nM IC50:  76.9nMAssay Description:Activity test of serotonin 5-HT6 receptor antagonists of the general formulas 1, 2 in the setting of competitive binding to serotonin 5-HT6 receptors...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM50396233(CHEMBL2172182 | US8569318, 1.1(3))
Affinity DataKi:  60nM IC50:  13nMAssay Description:Activity test of serotonin 5-HT6 receptor antagonists of the general formulas 1, 2 in the setting of competitive binding to serotonin 5-HT6 receptors...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM103946(CHEMBL2172189 | US8569318, 2.2(2))
Affinity DataKi:  372nM IC50:  801nMAssay Description:Activity test of serotonin 5-HT6 receptor antagonists of the general formulas 1, 2 in the setting of competitive binding to serotonin 5-HT6 receptors...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
TBA

US Patent
LigandPNGBDBM103947(CHEMBL2172190 | US8569318, 2.2(3))
Affinity DataIC50: >1.00E+3nMAssay Description:Activity test of serotonin 5-HT6 receptor antagonists of the general formulas 1, 2 in the setting of competitive binding to serotonin 5-HT6 receptors...More data for this Ligand-Target Pair
In DepthDetails US Patent