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Found 5 Enz. Inhib. hit(s) with all data for entry = 6068
TargetMAP/microtubule affinity-regulating kinase 3(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM107109(US8592425, 8)
Affinity DataIC50:  0.5nMAssay Description:MARK3 activity was assayed in vitro using a Cdc25C biotinylated peptide substrate (Cell Signalling Technologies). The phosphopeptide product was quan...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP/microtubule affinity-regulating kinase 3(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM107110(US8592425, 14)
Affinity DataIC50:  15nMAssay Description:MARK3 activity was assayed in vitro using a Cdc25C biotinylated peptide substrate (Cell Signalling Technologies). The phosphopeptide product was quan...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP/microtubule affinity-regulating kinase 3(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM107108(US8592425, 1)
Affinity DataIC50:  20nMAssay Description:MARK3 activity was assayed in vitro using a Cdc25C biotinylated peptide substrate (Cell Signalling Technologies). The phosphopeptide product was quan...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP/microtubule affinity-regulating kinase 3(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM107111(US8592425, 24)
Affinity DataIC50:  140nMAssay Description:MARK3 activity was assayed in vitro using a Cdc25C biotinylated peptide substrate (Cell Signalling Technologies). The phosphopeptide product was quan...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMAP/microtubule affinity-regulating kinase 3(Homo sapiens (Human))
Merck Sharp & Dohme

US Patent
LigandPNGBDBM107107(US8592425, 92)
Affinity DataIC50:  720nMAssay Description:MARK3 activity was assayed in vitro using a Cdc25C biotinylated peptide substrate (Cell Signalling Technologies). The phosphopeptide product was quan...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent