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Found 13 Enz. Inhib. hit(s) with all data for entry = 6166
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Tufts University

US Patent
LigandPNGBDBM112790(US8628961, PIT-7)
Affinity DataIC50:  1.34E+4nMpH: 7.5 T: 2°CAssay Description:In order to identify compounds that disrupt the interaction between PIP3 and PH domains, a high-throughput fluorescence polarization (FP)-binding ass...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Tufts University

US Patent
LigandPNGBDBM112786(US8628961, PIT-3)
Affinity DataIC50:  1.75E+4nMpH: 7.5 T: 2°CAssay Description:In order to identify compounds that disrupt the interaction between PIP3 and PH domains, a high-throughput fluorescence polarization (FP)-binding ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Tufts University

US Patent
LigandPNGBDBM112789(US8628961, PIT-6)
Affinity DataIC50:  1.81E+4nMpH: 7.5 T: 2°CAssay Description:In order to identify compounds that disrupt the interaction between PIP3 and PH domains, a high-throughput fluorescence polarization (FP)-binding ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Tufts University

US Patent
LigandPNGBDBM112788(US8628961, PIT-5)
Affinity DataIC50:  2.08E+4nMpH: 7.5 T: 2°CAssay Description:In order to identify compounds that disrupt the interaction between PIP3 and PH domains, a high-throughput fluorescence polarization (FP)-binding ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Tufts University

US Patent
LigandPNGBDBM112787(US8628961, PIT-4)
Affinity DataIC50:  2.26E+4nMpH: 7.5 T: 2°CAssay Description:In order to identify compounds that disrupt the interaction between PIP3 and PH domains, a high-throughput fluorescence polarization (FP)-binding ass...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Tufts University

US Patent
LigandPNGBDBM112785(US8628961, DM-PIT-1)
Affinity DataIC50:  2.71E+4nMpH: 7.5 T: 2°CAssay Description:In order to identify compounds that disrupt the interaction between PIP3 and PH domains, a high-throughput fluorescence polarization (FP)-binding ass...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Tufts University

US Patent
LigandPNGBDBM112784(US8628961, PIT-1)
Affinity DataIC50:  3.10E+4nMpH: 7.5 T: 2°CAssay Description:In order to identify compounds that disrupt the interaction between PIP3 and PH domains, a high-throughput fluorescence polarization (FP)-binding ass...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCytohesin-3(Homo sapiens (Human))
Tufts University

US Patent
LigandPNGBDBM112785(US8628961, DM-PIT-1)
Affinity DataIC50:  3.55E+4nMpH: 7.5 T: 2°CAssay Description:In order to identify compounds that disrupt the interaction between PIP3 and PH domains, a high-throughput fluorescence polarization (FP)-binding ass...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCytohesin-3(Homo sapiens (Human))
Tufts University

US Patent
LigandPNGBDBM112784(US8628961, PIT-1)
Affinity DataIC50:  4.03E+4nMpH: 7.5 T: 2°CAssay Description:In order to identify compounds that disrupt the interaction between PIP3 and PH domains, a high-throughput fluorescence polarization (FP)-binding ass...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Tufts University

US Patent
LigandPNGBDBM112790(US8628961, PIT-7)
Affinity DataIC50:  5.23E+4nMpH: 7.5 T: 2°CAssay Description:In order to identify compounds that disrupt the interaction between PIP3 and PH domains, a high-throughput fluorescence polarization (FP)-binding ass...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Tufts University

US Patent
LigandPNGBDBM112784(US8628961, PIT-1)
Affinity DataIC50:  6.67E+4nMpH: 7.5 T: 2°CAssay Description:In order to identify compounds that disrupt the interaction between PIP3 and PH domains, a high-throughput fluorescence polarization (FP)-binding ass...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Tufts University

US Patent
LigandPNGBDBM112785(US8628961, DM-PIT-1)
Affinity DataIC50:  8.05E+4nMpH: 7.5 T: 2°CAssay Description:In order to identify compounds that disrupt the interaction between PIP3 and PH domains, a high-throughput fluorescence polarization (FP)-binding ass...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Tufts University

US Patent
LigandPNGBDBM112786(US8628961, PIT-3)
Affinity DataIC50:  1.07E+5nMpH: 7.5 T: 2°CAssay Description:In order to identify compounds that disrupt the interaction between PIP3 and PH domains, a high-throughput fluorescence polarization (FP)-binding ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent