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Found 37 Enz. Inhib. hit(s) with all data for entry = 6328
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
The Ohio State University Research Foundation

US Patent
LigandPNGBDBM50430629(CHEMBL2332031 | US8741944, 71)
Affinity DataIC50:  2.00E+3nMAssay Description:PDK-1 kinase activity This in vitro assay was performed using a PDK-1 kinase assay kit (Upstate, Lake Placid, N.Y.) according to the vendor's ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
The Ohio State University Research Foundation

US Patent
LigandPNGBDBM50430630(CHEMBL1650595 | US8741944, 70)
Affinity DataIC50:  5.00E+3nMAssay Description:PDK-1 kinase activity This in vitro assay was performed using a PDK-1 kinase assay kit (Upstate, Lake Placid, N.Y.) according to the vendor's ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
The Ohio State University Research Foundation

US Patent
LigandPNGBDBM123427(US8741944, 49)
Affinity DataIC50:  9.00E+3nMAssay Description:PDK-1 kinase activity This in vitro assay was performed using a PDK-1 kinase assay kit (Upstate, Lake Placid, N.Y.) according to the vendor's ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
The Ohio State University Research Foundation

US Patent
LigandPNGBDBM123437(US8741944, 59)
Affinity DataIC50:  9.00E+3nMAssay Description:PDK-1 kinase activity This in vitro assay was performed using a PDK-1 kinase assay kit (Upstate, Lake Placid, N.Y.) according to the vendor's ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
The Ohio State University Research Foundation

US Patent
LigandPNGBDBM123439(US8741944, 61)
Affinity DataIC50:  1.20E+4nMAssay Description:PDK-1 kinase activity This in vitro assay was performed using a PDK-1 kinase assay kit (Upstate, Lake Placid, N.Y.) according to the vendor's ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
The Ohio State University Research Foundation

US Patent
LigandPNGBDBM123436(US8741944, 58)
Affinity DataIC50:  1.20E+4nMAssay Description:PDK-1 kinase activity This in vitro assay was performed using a PDK-1 kinase assay kit (Upstate, Lake Placid, N.Y.) according to the vendor's ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
The Ohio State University Research Foundation

US Patent
LigandPNGBDBM123434(US8741944, 56)
Affinity DataIC50:  1.50E+4nMAssay Description:PDK-1 kinase activity This in vitro assay was performed using a PDK-1 kinase assay kit (Upstate, Lake Placid, N.Y.) according to the vendor's ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
The Ohio State University Research Foundation

US Patent
LigandPNGBDBM123428(US8741944, 50)
Affinity DataIC50:  1.50E+4nMAssay Description:PDK-1 kinase activity This in vitro assay was performed using a PDK-1 kinase assay kit (Upstate, Lake Placid, N.Y.) according to the vendor's ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
The Ohio State University Research Foundation

US Patent
LigandPNGBDBM123446(US8741944, 68)
Affinity DataIC50:  1.50E+4nMAssay Description:PDK-1 kinase activity This in vitro assay was performed using a PDK-1 kinase assay kit (Upstate, Lake Placid, N.Y.) according to the vendor's ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
The Ohio State University Research Foundation

US Patent
LigandPNGBDBM123444(US8741944, 66)
Affinity DataIC50:  1.60E+4nMAssay Description:PDK-1 kinase activity This in vitro assay was performed using a PDK-1 kinase assay kit (Upstate, Lake Placid, N.Y.) according to the vendor's ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
The Ohio State University Research Foundation

US Patent
LigandPNGBDBM123435(US8741944, 57)
Affinity DataIC50:  1.60E+4nMAssay Description:PDK-1 kinase activity This in vitro assay was performed using a PDK-1 kinase assay kit (Upstate, Lake Placid, N.Y.) according to the vendor's ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
The Ohio State University Research Foundation

US Patent
LigandPNGBDBM123431(US8741944, 53)
Affinity DataIC50:  1.70E+4nMAssay Description:PDK-1 kinase activity This in vitro assay was performed using a PDK-1 kinase assay kit (Upstate, Lake Placid, N.Y.) according to the vendor's ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
The Ohio State University Research Foundation

US Patent
LigandPNGBDBM123425(US8741944, 47)
Affinity DataIC50:  1.80E+4nMAssay Description:PDK-1 kinase activity This in vitro assay was performed using a PDK-1 kinase assay kit (Upstate, Lake Placid, N.Y.) according to the vendor's ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
The Ohio State University Research Foundation

US Patent
LigandPNGBDBM123429(US8741944, 51)
Affinity DataIC50:  1.80E+4nMAssay Description:PDK-1 kinase activity This in vitro assay was performed using a PDK-1 kinase assay kit (Upstate, Lake Placid, N.Y.) according to the vendor's ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
The Ohio State University Research Foundation

US Patent
LigandPNGBDBM123430(US8741944, 52)
Affinity DataIC50:  2.00E+4nMAssay Description:PDK-1 kinase activity This in vitro assay was performed using a PDK-1 kinase assay kit (Upstate, Lake Placid, N.Y.) according to the vendor's ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
The Ohio State University Research Foundation

US Patent
LigandPNGBDBM123420(US8741944, 41)
Affinity DataIC50:  2.00E+4nMAssay Description:PDK-1 kinase activity This in vitro assay was performed using a PDK-1 kinase assay kit (Upstate, Lake Placid, N.Y.) according to the vendor's ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
The Ohio State University Research Foundation

US Patent
LigandPNGBDBM123423(US8741944, 45)
Affinity DataIC50:  2.10E+4nMAssay Description:PDK-1 kinase activity This in vitro assay was performed using a PDK-1 kinase assay kit (Upstate, Lake Placid, N.Y.) according to the vendor's ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
The Ohio State University Research Foundation

US Patent
LigandPNGBDBM123424(US8741944, 46)
Affinity DataIC50:  2.20E+4nMAssay Description:PDK-1 kinase activity This in vitro assay was performed using a PDK-1 kinase assay kit (Upstate, Lake Placid, N.Y.) according to the vendor's ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
The Ohio State University Research Foundation

US Patent
LigandPNGBDBM123426(US8741944, 48)
Affinity DataIC50:  2.30E+4nMAssay Description:PDK-1 kinase activity This in vitro assay was performed using a PDK-1 kinase assay kit (Upstate, Lake Placid, N.Y.) according to the vendor's ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
The Ohio State University Research Foundation

US Patent
LigandPNGBDBM123422(US8741944, 43)
Affinity DataIC50:  2.40E+4nMAssay Description:PDK-1 kinase activity This in vitro assay was performed using a PDK-1 kinase assay kit (Upstate, Lake Placid, N.Y.) according to the vendor's ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
The Ohio State University Research Foundation

US Patent
LigandPNGBDBM123443(US8741944, 65)
Affinity DataIC50:  2.50E+4nMAssay Description:PDK-1 kinase activity This in vitro assay was performed using a PDK-1 kinase assay kit (Upstate, Lake Placid, N.Y.) according to the vendor's ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
The Ohio State University Research Foundation

US Patent
LigandPNGBDBM123433(US8741944, 55)
Affinity DataIC50:  3.20E+4nMAssay Description:PDK-1 kinase activity This in vitro assay was performed using a PDK-1 kinase assay kit (Upstate, Lake Placid, N.Y.) according to the vendor's ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
The Ohio State University Research Foundation

US Patent
LigandPNGBDBM123418(US8741944, 39)
Affinity DataIC50:  3.20E+4nMAssay Description:PDK-1 kinase activity This in vitro assay was performed using a PDK-1 kinase assay kit (Upstate, Lake Placid, N.Y.) according to the vendor's ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
The Ohio State University Research Foundation

US Patent
LigandPNGBDBM123432(US8741944, 54)
Affinity DataIC50:  3.20E+4nMAssay Description:PDK-1 kinase activity This in vitro assay was performed using a PDK-1 kinase assay kit (Upstate, Lake Placid, N.Y.) according to the vendor's ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
The Ohio State University Research Foundation

US Patent
LigandPNGBDBM123419(US8741944, 40)
Affinity DataIC50:  3.40E+4nMAssay Description:PDK-1 kinase activity This in vitro assay was performed using a PDK-1 kinase assay kit (Upstate, Lake Placid, N.Y.) according to the vendor's ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
The Ohio State University Research Foundation

US Patent
LigandPNGBDBM123421(US8741944, 42)
Affinity DataIC50:  3.40E+4nMAssay Description:PDK-1 kinase activity This in vitro assay was performed using a PDK-1 kinase assay kit (Upstate, Lake Placid, N.Y.) according to the vendor's ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
The Ohio State University Research Foundation

US Patent
LigandPNGBDBM123417(US8741944, 38)
Affinity DataIC50:  3.80E+4nMAssay Description:PDK-1 kinase activity This in vitro assay was performed using a PDK-1 kinase assay kit (Upstate, Lake Placid, N.Y.) according to the vendor's ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
The Ohio State University Research Foundation

US Patent
LigandPNGBDBM123441(US8741944, 63)
Affinity DataIC50:  4.00E+4nMAssay Description:PDK-1 kinase activity This in vitro assay was performed using a PDK-1 kinase assay kit (Upstate, Lake Placid, N.Y.) according to the vendor's ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
The Ohio State University Research Foundation

US Patent
LigandPNGBDBM123448(US8741944, 72)
Affinity DataIC50:  4.00E+4nMAssay Description:PDK-1 kinase activity This in vitro assay was performed using a PDK-1 kinase assay kit (Upstate, Lake Placid, N.Y.) according to the vendor's ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
The Ohio State University Research Foundation

US Patent
LigandPNGBDBM123445(US8741944, 67)
Affinity DataIC50:  4.20E+4nMAssay Description:PDK-1 kinase activity This in vitro assay was performed using a PDK-1 kinase assay kit (Upstate, Lake Placid, N.Y.) according to the vendor's ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
The Ohio State University Research Foundation

US Patent
LigandPNGBDBM123416(US8741944, 37)
Affinity DataIC50:  4.20E+4nMAssay Description:PDK-1 kinase activity This in vitro assay was performed using a PDK-1 kinase assay kit (Upstate, Lake Placid, N.Y.) according to the vendor's ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
The Ohio State University Research Foundation

US Patent
LigandPNGBDBM123438(US8741944, 60)
Affinity DataIC50:  4.20E+4nMAssay Description:PDK-1 kinase activity This in vitro assay was performed using a PDK-1 kinase assay kit (Upstate, Lake Placid, N.Y.) according to the vendor's ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
The Ohio State University Research Foundation

US Patent
LigandPNGBDBM123440(US8741944, 62)
Affinity DataIC50:  4.50E+4nMAssay Description:PDK-1 kinase activity This in vitro assay was performed using a PDK-1 kinase assay kit (Upstate, Lake Placid, N.Y.) according to the vendor's ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
The Ohio State University Research Foundation

US Patent
LigandPNGBDBM123447(US8741944, 69)
Affinity DataIC50:  4.50E+4nMAssay Description:PDK-1 kinase activity This in vitro assay was performed using a PDK-1 kinase assay kit (Upstate, Lake Placid, N.Y.) according to the vendor's ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
The Ohio State University Research Foundation

US Patent
LigandPNGBDBM11639(4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyraz...)
Affinity DataIC50:  4.80E+4nMAssay Description:PDK-1 kinase activity This in vitro assay was performed using a PDK-1 kinase assay kit (Upstate, Lake Placid, N.Y.) according to the vendor's ins...More data for this Ligand-Target Pair
In DepthDetails US PatentDrugBank

Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
The Ohio State University Research Foundation

US Patent
LigandPNGBDBM123442(US8741944, 64)
Affinity DataIC50:  5.20E+4nMAssay Description:PDK-1 kinase activity This in vitro assay was performed using a PDK-1 kinase assay kit (Upstate, Lake Placid, N.Y.) according to the vendor's ins...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
The Ohio State University Research Foundation

US Patent
LigandPNGBDBM50376854(CHEMBL261143 | US8741944, 44)
Affinity DataIC50:  6.50E+4nMAssay Description:PDK-1 kinase activity This in vitro assay was performed using a PDK-1 kinase assay kit (Upstate, Lake Placid, N.Y.) according to the vendor's ins...More data for this Ligand-Target Pair
In DepthDetails US Patent