Compile Data Set for Download or QSAR
maximum 50k data
Found 20 Enz. Inhib. hit(s) with all data for entry = 6389
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Kyoto University

US Patent
LigandPNGBDBM125988(US8772297, Y244)
Affinity DataIC50:  600nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Kyoto University

US Patent
LigandPNGBDBM125985(US8772297, Y241)
Affinity DataIC50:  700nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Kyoto University

US Patent
LigandPNGBDBM125986(US8772297, Y260)
Affinity DataIC50:  1.50E+3nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Kyoto University

US Patent
LigandPNGBDBM125979(US8772297, Y177)
Affinity DataIC50:  2.00E+3nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Kyoto University

US Patent
LigandPNGBDBM125980(US8772297, Y224)
Affinity DataIC50:  2.40E+3nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Kyoto University

US Patent
LigandPNGBDBM125989(US8772297, Y250)
Affinity DataIC50:  2.50E+3nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Kyoto University

US Patent
LigandPNGBDBM125981(US8772297, Y186)
Affinity DataIC50:  3.60E+3nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Kyoto University

US Patent
LigandPNGBDBM125991(US8772297, Y296)
Affinity DataIC50:  4.60E+3nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Kyoto University

US Patent
LigandPNGBDBM125990(US8772297, Y284)
Affinity DataIC50:  6.70E+3nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Kyoto University

US Patent
LigandPNGBDBM125987(US8772297, Y366)
Affinity DataIC50:  7.30E+3nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Kyoto University

US Patent
LigandPNGBDBM125976(US8772297, Y145)
Affinity DataIC50:  8.00E+3nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Kyoto University

US Patent
LigandPNGBDBM125978(US8772297, Y155)
Affinity DataIC50:  1.40E+4nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Kyoto University

US Patent
LigandPNGBDBM125982(US8772297, Y178)
Affinity DataIC50:  1.50E+4nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Kyoto University

US Patent
LigandPNGBDBM125984(US8772297, Y196)
Affinity DataIC50:  1.60E+4nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Kyoto University

US Patent
LigandPNGBDBM125973(US8772297, Y141)
Affinity DataIC50:  1.70E+4nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Kyoto University

US Patent
LigandPNGBDBM125977(US8772297, Y147)
Affinity DataIC50:  1.80E+4nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Kyoto University

US Patent
LigandPNGBDBM125974(US8772297, Y142)
Affinity DataIC50:  2.20E+4nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Kyoto University

US Patent
LigandPNGBDBM125983(US8772297, Y185)
Affinity DataIC50:  2.40E+4nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Kyoto University

US Patent
LigandPNGBDBM125972(US8772297, Y098)
Affinity DataIC50:  2.70E+4nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetTGF-beta receptor type-1(Homo sapiens (Human))
Kyoto University

US Patent
LigandPNGBDBM125975(US8772297, Y140)
Affinity DataIC50:  3.00E+4nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In DepthDetails US Patent