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Found 12 Enz. Inhib. hit(s) with all data for entry = 6516
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Development Center For Biotechnology

US Patent
LigandPNGBDBM135802(US8853207, Example-82)
Affinity DataIC50:  12.2nMAssay Description:Inhibition of C-kit kinase activity by compounds disclosed herein was quantified by measuring the amount of [33P] incorporated into the substrate in ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Development Center For Biotechnology

US Patent
LigandPNGBDBM135799(US8853207, Example-69)
Affinity DataIC50:  22nMAssay Description:Inhibition of C-kit kinase activity by compounds disclosed herein was quantified by measuring the amount of [33P] incorporated into the substrate in ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Development Center For Biotechnology

US Patent
LigandPNGBDBM135800(US8853207, Example-70)
Affinity DataIC50:  24.8nMAssay Description:Inhibition of C-kit kinase activity by compounds disclosed herein was quantified by measuring the amount of [33P] incorporated into the substrate in ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Development Center For Biotechnology

US Patent
LigandPNGBDBM135801(US8853207, Example-78)
Affinity DataIC50:  27.5nMAssay Description:Inhibition of C-kit kinase activity by compounds disclosed herein was quantified by measuring the amount of [33P] incorporated into the substrate in ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Development Center For Biotechnology

US Patent
LigandPNGBDBM135798(US8853207, Example-10)
Affinity DataIC50:  118nMpH: 7.0Assay Description:Inhibition of PDGFR-beta kinase activity by compounds disclosed herein was quantified by measuring the amount of [33P] incorporated into the substrat...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Development Center For Biotechnology

US Patent
LigandPNGBDBM135798(US8853207, Example-10)
Affinity DataIC50:  139nMAssay Description:Inhibition of C-kit kinase activity by compounds disclosed herein was quantified by measuring the amount of [33P] incorporated into the substrate in ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Development Center For Biotechnology

US Patent
LigandPNGBDBM135802(US8853207, Example-82)
Affinity DataIC50:  176nMpH: 7.0Assay Description:Inhibition of PDGFR-beta kinase activity by compounds disclosed herein was quantified by measuring the amount of [33P] incorporated into the substrat...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMast/stem cell growth factor receptor Kit(Homo sapiens (Human))
Development Center For Biotechnology

US Patent
LigandPNGBDBM135797(US8853207, Example-2)
Affinity DataIC50:  201nMAssay Description:Inhibition of C-kit kinase activity by compounds disclosed herein was quantified by measuring the amount of [33P] incorporated into the substrate in ...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Development Center For Biotechnology

US Patent
LigandPNGBDBM135799(US8853207, Example-69)
Affinity DataIC50:  316nMpH: 7.0Assay Description:Inhibition of PDGFR-beta kinase activity by compounds disclosed herein was quantified by measuring the amount of [33P] incorporated into the substrat...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Development Center For Biotechnology

US Patent
LigandPNGBDBM135801(US8853207, Example-78)
Affinity DataIC50:  363nMpH: 7.0Assay Description:Inhibition of PDGFR-beta kinase activity by compounds disclosed herein was quantified by measuring the amount of [33P] incorporated into the substrat...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Development Center For Biotechnology

US Patent
LigandPNGBDBM135800(US8853207, Example-70)
Affinity DataIC50:  479nMpH: 7.0Assay Description:Inhibition of PDGFR-beta kinase activity by compounds disclosed herein was quantified by measuring the amount of [33P] incorporated into the substrat...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Development Center For Biotechnology

US Patent
LigandPNGBDBM135797(US8853207, Example-2)
Affinity DataIC50:  859nMpH: 7.0Assay Description:Inhibition of PDGFR-beta kinase activity by compounds disclosed herein was quantified by measuring the amount of [33P] incorporated into the substrat...More data for this Ligand-Target Pair
In DepthDetails US Patent