Compile Data Set for Download or QSAR
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Found 10 Enz. Inhib. hit(s) with all data for entry = 7032
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM167874(US9073925, 3)
Affinity DataKi:  5.90nM ΔG°:  -47.0kJ/molepH: 7.4 T: 2°CAssay Description:Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM167873(US9073925, 2)
Affinity DataKi:  6.40nM ΔG°:  -46.8kJ/molepH: 7.4 T: 2°CAssay Description:Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM167878(US9073925, 7)
Affinity DataKi:  11nM ΔG°:  -45.4kJ/molepH: 7.4 T: 2°CAssay Description:Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM167880(US9073925, 9)
Affinity DataKi:  15nM ΔG°:  -44.7kJ/molepH: 7.4 T: 2°CAssay Description:Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM167881(US9073925, 10)
Affinity DataKi:  15nM ΔG°:  -44.7kJ/molepH: 7.4 T: 2°CAssay Description:Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM167876(US9073925, 5)
Affinity DataKi:  23nM ΔG°:  -43.6kJ/molepH: 7.4 T: 2°CAssay Description:Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM167882(US9073925, 11)
Affinity DataKi:  25nM ΔG°:  -43.4kJ/molepH: 7.4 T: 2°CAssay Description:Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM167879(US9073925, 8)
Affinity DataKi:  29nM ΔG°:  -43.0kJ/molepH: 7.4 T: 2°CAssay Description:Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM167875(US9073925, 4)
Affinity DataKi:  44nM ΔG°:  -42.0kJ/molepH: 7.4 T: 2°CAssay Description:Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM167877(US9073925, 6)
Affinity DataKi:  123nM ΔG°:  -39.4kJ/molepH: 7.4 T: 2°CAssay Description:Evaluation of the affinity of compounds for the human MCH-1 receptor was accomplished using 4-(3,4,5-tritritiumbenzyloxy)-1-(1-(2-(pyrrolidin-1-yl)et...More data for this Ligand-Target Pair
In DepthDetails US Patent