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Found 4 Enz. Inhib. hit(s) with all data for entry = 8039
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM230879(US9346822, 41)
Affinity DataIC50:  0.100nMAssay Description:The monkey and human membrane fractions prepared were diluted with the assay buffer to yield a 200 g/ml dilution, each of which was then dispensed at...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Takeda Pharmaceutical

US Patent
LigandPNGBDBM50347988(CHEMBL1800152 | US9346822, 40)
Affinity DataIC50:  0.200nMAssay Description:The monkey and human membrane fractions prepared were diluted with the assay buffer to yield a 200 g/ml dilution, each of which was then dispensed at...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGonadotropin-releasing hormone receptor(Macaca fascicularis (Crab-eating macaque) (Cynomol...)
Takeda Pharmaceutical

US Patent
LigandPNGBDBM230879(US9346822, 41)
Affinity DataIC50:  3nMAssay Description:The monkey and human membrane fractions prepared were diluted with the assay buffer to yield a 200 g/ml dilution, each of which was then dispensed at...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGonadotropin-releasing hormone receptor(Macaca fascicularis (Crab-eating macaque) (Cynomol...)
Takeda Pharmaceutical

US Patent
LigandPNGBDBM50347988(CHEMBL1800152 | US9346822, 40)
Affinity DataIC50:  9nMAssay Description:The monkey and human membrane fractions prepared were diluted with the assay buffer to yield a 200 g/ml dilution, each of which was then dispensed at...More data for this Ligand-Target Pair
In DepthDetails US Patent