Compile Data Set for Download or QSAR
maximum 50k data
Found 68 Enz. Inhib. hit(s) with all data for entry = 997
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179693(US9127001, 8b | US9598410, Compound 8b)
Affinity DataIC50:  19nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179694(US9127001, 8c | US9598410, Compound 8c)
Affinity DataIC50:  47nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179702(US9127001, 8i | US9598410, Compound 8i)
Affinity DataIC50:  64nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179635(US9127001, 6n | US9598410, Compound 6n)
Affinity DataIC50:  91nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179623(US9127001, 6a | US9598410, Compound 6a)
Affinity DataIC50:  95nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179629(US9127001, 6g | US9598410, Compound 6g)
Affinity DataIC50:  99.5nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179659(US9127001, 6am | US9598410, Compound 6am)
Affinity DataIC50:  114nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179708(US9127001, 8o | US9598410, Compound 8o)
Affinity DataIC50:  131nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179624(US9127001, 6b | US9598410, Compound 6b)
Affinity DataIC50:  172nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179660(US9127001, 6an | US9598410, Compound 6an)
Affinity DataIC50:  187nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179630(US9127001, 6h | US9598410, Compound 6h)
Affinity DataIC50:  190nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179625(US9127001, 6c | US9598410, Compound 6c)
Affinity DataIC50:  215nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179631(US9127001, 6i | US9598410, Compound 6i)
Affinity DataIC50:  216nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179713(US9127001, 8t | US9598410, Compound 8t)
Affinity DataIC50:  246nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179683(US9127001, 6bl | US9127001, 6bm | US9598410, Compo...)
Affinity DataIC50:  251nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179661(US9127001, 6ao | US9598410, Compound 6ao)
Affinity DataIC50:  258nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179657(US9127001, 6ak | US9598410, Compound 6ak)
Affinity DataIC50:  270nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179692(US9127001, 8a | US9598410, Compound 8a)
Affinity DataIC50:  276nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179662(US9127001, 6ap | US9598410, Compound 6ap)
Affinity DataIC50:  285nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179663(US9127001, 6aq | US9598410, Compound 6aq)
Affinity DataIC50:  359nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179725(US9127001, 12a | US9598410, Compound 12a)
Affinity DataIC50:  380nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179678(US9127001, 6bg | US9598410, Compound 6bg)
Affinity DataIC50:  398nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179714(US9127001, 8u | US9598410, Compound 8u)
Affinity DataIC50:  416nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179730(US9127001, 13a | US9598410, Compound 13a)
Affinity DataIC50:  422nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179626(US9127001, 6d | US9598410, Compound 6d)
Affinity DataIC50:  422nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179731(US9127001, 13b | US9598410, Compound 13b)
Affinity DataIC50:  462nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179664(US9127001, 6ar | US9127001, 6be | US9127001, 6bf |...)
Affinity DataIC50:  500nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179664(US9127001, 6ar | US9127001, 6be | US9127001, 6bf |...)
Affinity DataIC50:  500nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179697(US9127001, 8z | US9598410, Compound 8z)
Affinity DataIC50:  511nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179726(US9127001, 12b | US9598410, Compound 12b)
Affinity DataIC50:  511nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179709(US9127001, 8p | US9598410, Compound 8p)
Affinity DataIC50:  530nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM302143(3-(4-Fluoro-phenyl)-1-[(R)-1-(4-fluoro-phenyl)-eth...)
Affinity DataIC50:  540nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179664(US9127001, 6ar | US9127001, 6be | US9127001, 6bf |...)
Affinity DataIC50:  552nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179705(US9127001, 8l | US9598410, Compound 8l)
Affinity DataIC50:  585nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179628(US9127001, 6f | US9598410, Compound 6f)
Affinity DataIC50:  598nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM302144(3-(4-Fluoro-phenyl)-1-[(R)-1-(4-fluoro-phenyl)-eth...)
Affinity DataIC50:  611nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179665(US9127001, 6as | US9598410, Compound 6as)
Affinity DataIC50:  659nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179666(US9127001, 6at | US9598410, Compound 6at)
Affinity DataIC50:  720nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179703(US9127001, 8j | US9598410, Compound 8j)
Affinity DataIC50:  722nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179727(US9127001, 12c | US9598410, Compound 12c)
Affinity DataIC50:  734nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179710(US9127001, 8q | US9598410, Compound 8q)
Affinity DataIC50:  756nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179715(US9127001, 8v | US9598410, Compound 8v)
Affinity DataIC50:  864nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179706(US9127001, 8m | US9598410, Compound 8m)
Affinity DataIC50:  890nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179704(US9127001, 8k | US9598410, Compound 8k)
Affinity DataIC50:  906nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179667(US9127001, 6av | US9598410, Compound 6av)
Affinity DataIC50:  911nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179668(US9127001, 6aw | US9598410, Compound 6aw)
Affinity DataIC50:  947nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179683(US9127001, 6bl | US9127001, 6bm | US9598410, Compo...)
Affinity DataIC50:  966nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179669(US9127001, 6ax | US9598410, Compound 6ax)
Affinity DataIC50:  975nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179711(US9127001, 8r | US9598410, Compound 8r)
Affinity DataIC50:  1.14E+3nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetPotassium channel subfamily K member 3(Homo sapiens (Human))
Sanofi

US Patent
LigandPNGBDBM179696(US9127001, 8w | US9598410, Compound 8w)
Affinity DataIC50:  1.15E+3nMAssay Description:Human TASK-1 channels were expressed in Xenopus oocytes. For this purpose, oocytes were isolated from Xenopus laevis and defoliated. Subsequently, TA...More data for this Ligand-Target Pair
In DepthDetails US Patent
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