Compile Data Set for Download or QSAR
maximum 50k data
Found 12 Enz. Inhib. hit(s) with all data for entry = 32
TargetBile acid receptor(Homo sapiens (Human))
Albireo

US Patent
LigandPNGBDBM77055(US10093697, 8. | US10487111, Example 8. | US969401...)
Affinity DataIC50:  0.110nMAssay Description:ISBT Hu HEK Uptake SPA 13203 IBAT HUM Ileal Bile Acid Transporter Human HEK Glycocholic acid Uptake Radiometric¿SPA Inhibitor IC50 Mean IC50 (nM) was...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBile acid receptor(Homo sapiens (Human))
Albireo

US Patent
LigandPNGBDBM77086(US10093697, 13. | US10487111, Example 13. | US9694...)
Affinity DataIC50:  0.130nMAssay Description:ISBT Hu HEK Uptake SPA 13203 IBAT HUM Ileal Bile Acid Transporter Human HEK Glycocholic acid Uptake Radiometric¿SPA Inhibitor IC50 Mean IC50 (nM) was...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBile acid receptor(Homo sapiens (Human))
Albireo

US Patent
LigandPNGBDBM77080(US10093697, 11. | US9694018, 11)
Affinity DataIC50:  0.150nMAssay Description:ISBT Hu HEK Uptake SPA 13203 IBAT HUM Ileal Bile Acid Transporter Human HEK Glycocholic acid Uptake Radiometric¿SPA Inhibitor IC50 Mean IC50 (nM) was...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBile acid receptor(Homo sapiens (Human))
Albireo

US Patent
LigandPNGBDBM77040(US10093697, 5. | US10487111, Example 5. | US969401...)
Affinity DataIC50:  0.160nMAssay Description:ISBT Hu HEK Uptake SPA 13203 IBAT HUM Ileal Bile Acid Transporter Human HEK Glycocholic acid Uptake Radiometric¿SPA Inhibitor IC50 Mean IC50 (nM) was...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBile acid receptor(Homo sapiens (Human))
Albireo

US Patent
LigandPNGBDBM77029(US10093697, 3. | US10487111, Example 3. | US969401...)
Affinity DataIC50:  0.180nMAssay Description:ISBT Hu HEK Uptake SPA 13203 IBAT HUM Ileal Bile Acid Transporter Human HEK Glycocholic acid Uptake Radiometric¿SPA Inhibitor IC50 Mean IC50 (nM) was...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBile acid receptor(Homo sapiens (Human))
Albireo

US Patent
LigandPNGBDBM77074(US10093697, 10. | US10487111, Example 10. | US9694...)
Affinity DataIC50:  0.200nMAssay Description:ISBT Hu HEK Uptake SPA 13203 IBAT HUM Ileal Bile Acid Transporter Human HEK Glycocholic acid Uptake Radiometric¿SPA Inhibitor IC50 Mean IC50 (nM) was...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBile acid receptor(Homo sapiens (Human))
Albireo

US Patent
LigandPNGBDBM77083(US10093697, 12. | US10487111, Example 12. | US9694...)
Affinity DataIC50:  0.300nMAssay Description:ISBT Hu HEK Uptake SPA 13203 IBAT HUM Ileal Bile Acid Transporter Human HEK Glycocholic acid Uptake Radiometric¿SPA Inhibitor IC50 Mean IC50 (nM) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBile acid receptor(Homo sapiens (Human))
Albireo

US Patent
LigandPNGBDBM77033(US10093697, 4. | US10487111, Example 4. | US969401...)
Affinity DataIC50:  0.350nMAssay Description:ISBT Hu HEK Uptake SPA 13203 IBAT HUM Ileal Bile Acid Transporter Human HEK Glycocholic acid Uptake Radiometric¿SPA Inhibitor IC50 Mean IC50 (nM) was...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBile acid receptor(Homo sapiens (Human))
Albireo

US Patent
LigandPNGBDBM77051(US10093697, 7. | US10487111, Example 7. | US969401...)
Affinity DataIC50:  0.360nMAssay Description:ISBT Hu HEK Uptake SPA 13203 IBAT HUM Ileal Bile Acid Transporter Human HEK Glycocholic acid Uptake Radiometric¿SPA Inhibitor IC50 Mean IC50 (nM) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBile acid receptor(Homo sapiens (Human))
Albireo

US Patent
LigandPNGBDBM76996(US10487111, Example 2. | US9694018, 2)
Affinity DataIC50:  0.390nMAssay Description:ISBT Hu HEK Uptake SPA 13203 IBAT HUM Ileal Bile Acid Transporter Human HEK Glycocholic acid Uptake Radiometric¿SPA Inhibitor IC50 Mean IC50 (nM) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBile acid receptor(Homo sapiens (Human))
Albireo

US Patent
LigandPNGBDBM76994(US10093697, 1. | US10487111, Example 1. | US969401...)
Affinity DataIC50:  0.450nMAssay Description:ISBT Hu HEK Uptake SPA 13203 IBAT HUM Ileal Bile Acid Transporter Human HEK Glycocholic acid Uptake Radiometric¿SPA Inhibitor IC50 Mean IC50 (nM) was...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetBile acid receptor(Homo sapiens (Human))
Albireo

US Patent
LigandPNGBDBM77088(US10093697, 14. | US10487111, Example 14. | US9694...)
Affinity DataIC50:  1.20nMAssay Description:ISBT Hu HEK Uptake SPA 13203 IBAT HUM Ileal Bile Acid Transporter Human HEK Glycocholic acid Uptake Radiometric¿SPA Inhibitor IC50 Mean IC50 (nM) was...More data for this Ligand-Target Pair
In DepthDetails US Patent