Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with all data for entry = 2706
TargetProto-oncogene tyrosine-protein kinase receptor Ret [658-1114](Homo sapiens (Human))
Glaxosmithkline

US Patent
LigandPNGBDBM376389(N-(3-(2-(dimethylamino)ethoxy)-5-(trifluoromethyl)...)
Affinity DataIC50: <10nMAssay Description:Human RET kinase cytoplasmic domain (amino acids 658-1114 of accession number NP_000314.1) was expressed as an N-terminal GST-fusion protein using a ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetProto-oncogene tyrosine-protein kinase receptor Ret [658-1114](Homo sapiens (Human))
Glaxosmithkline

US Patent
LigandPNGBDBM376119(N-(2-(dimethylamino)ethyl)-3-(2-(4-(4-ethoxy-6-oxo...)
Affinity DataIC50: <10nMAssay Description:Human RET kinase cytoplasmic domain (amino acids 658-1114 of accession number NP_000314.1) was expressed as an N-terminal GST-fusion protein using a ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent