Compile Data Set for Download or QSAR
maximum 50k data
Found 11 Enz. Inhib. hit(s) with all data for entry = 3202
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Fondazione Istituto Itaiano Di Tecnologia

US Patent
LigandPNGBDBM394126(US9975861, 6)
Affinity DataIC50:  4.34E+3nMAssay Description:Human recombinant GSK-3β was purchased from Millipore (Millipore Iberica S.A.U.) The prephosphorylated polypeptide substrate was purchased from ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Fondazione Istituto Itaiano Di Tecnologia

US Patent
LigandPNGBDBM394127(US9975861, 9)
Affinity DataIC50:  6.93E+3nMAssay Description:Human recombinant GSK-3β was purchased from Millipore (Millipore Iberica S.A.U.) The prephosphorylated polypeptide substrate was purchased from ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Fondazione Istituto Itaiano Di Tecnologia

US Patent
LigandPNGBDBM394123(US9975861, 3 | US9975861, 4 | US9975861, 5)
Affinity DataIC50:  7.11E+3nMAssay Description:Human recombinant GSK-3β was purchased from Millipore (Millipore Iberica S.A.U.) The prephosphorylated polypeptide substrate was purchased from ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Fondazione Istituto Itaiano Di Tecnologia

US Patent
LigandPNGBDBM394123(US9975861, 3 | US9975861, 4 | US9975861, 5)
Affinity DataIC50:  8.13E+3nMAssay Description:β-secretase (BACE-1, Sigma-Aldrich) inhibition studies were performed by employing a peptide mimicking APP sequence as substrate (Methoxycoumari...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Fondazione Istituto Itaiano Di Tecnologia

US Patent
LigandPNGBDBM394123(US9975861, 3 | US9975861, 4 | US9975861, 5)
Affinity DataIC50:  1.26E+4nMAssay Description:β-secretase (BACE-1, Sigma-Aldrich) inhibition studies were performed by employing a peptide mimicking APP sequence as substrate (Methoxycoumari...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Fondazione Istituto Itaiano Di Tecnologia

US Patent
LigandPNGBDBM394123(US9975861, 3 | US9975861, 4 | US9975861, 5)
Affinity DataIC50:  1.26E+4nMAssay Description:Human recombinant GSK-3β was purchased from Millipore (Millipore Iberica S.A.U.) The prephosphorylated polypeptide substrate was purchased from ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Fondazione Istituto Itaiano Di Tecnologia

US Patent
LigandPNGBDBM394123(US9975861, 3 | US9975861, 4 | US9975861, 5)
Affinity DataIC50:  1.57E+4nMAssay Description:Human recombinant GSK-3β was purchased from Millipore (Millipore Iberica S.A.U.) The prephosphorylated polypeptide substrate was purchased from ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Fondazione Istituto Itaiano Di Tecnologia

US Patent
LigandPNGBDBM394123(US9975861, 3 | US9975861, 4 | US9975861, 5)
Affinity DataIC50:  1.61E+4nMAssay Description:β-secretase (BACE-1, Sigma-Aldrich) inhibition studies were performed by employing a peptide mimicking APP sequence as substrate (Methoxycoumari...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Fondazione Istituto Itaiano Di Tecnologia

US Patent
LigandPNGBDBM394126(US9975861, 6)
Affinity DataIC50:  3.68E+4nMAssay Description:β-secretase (BACE-1, Sigma-Aldrich) inhibition studies were performed by employing a peptide mimicking APP sequence as substrate (Methoxycoumari...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Fondazione Istituto Itaiano Di Tecnologia

US Patent
LigandPNGBDBM394122(US9975861, 2)
Affinity DataIC50:  4.07E+4nMAssay Description:Human recombinant GSK-3β was purchased from Millipore (Millipore Iberica S.A.U.) The prephosphorylated polypeptide substrate was purchased from ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetBeta-secretase 1(Homo sapiens (Human))
Fondazione Istituto Itaiano Di Tecnologia

US Patent
LigandPNGBDBM394122(US9975861, 2)
Affinity DataIC50:  5.03E+4nMAssay Description:β-secretase (BACE-1, Sigma-Aldrich) inhibition studies were performed by employing a peptide mimicking APP sequence as substrate (Methoxycoumari...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent