Compile Data Set for Download or QSAR
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Found 8 Enz. Inhib. hit(s) with all data for entry = 3313
TargetCannabinoid receptor 1(Mus musculus (Mouse))
Jenrin Discovery

US Patent
LigandPNGBDBM286106(US10617673, Example 4 | US11179370, Example 4 | US...)
Affinity DataIC50: >100nMAssay Description:Compound binding to CB1R was assessed in competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCannabinoid receptor 1(Mus musculus (Mouse))
Jenrin Discovery

US Patent
LigandPNGBDBM397087(US10617673, Example 2 | US11179370, Example 2 | US...)
Affinity DataIC50: >100nMAssay Description:Compound binding to CB1R was assessed in competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCannabinoid receptor 1(Mus musculus (Mouse))
Jenrin Discovery

US Patent
LigandPNGBDBM286100(US10617673, Example 1 | US11179370, Example 1 | US...)
Affinity DataIC50: >100nMAssay Description:Compound binding to CB1R was assessed in competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCannabinoid receptor 1(Mus musculus (Mouse))
Jenrin Discovery

US Patent
LigandPNGBDBM286104(US10617673, Example 3 | US11179370, Example 3 | US...)
Affinity DataIC50: >100nMAssay Description:Compound binding to CB1R was assessed in competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCannabinoid receptor 1(Mus musculus (Mouse))
Jenrin Discovery

US Patent
LigandPNGBDBM286105(US10617673, Example 3a (2S,4'R) | US11179370, Exam...)
Affinity DataIC50:  550nMAssay Description:Compound binding to CB1R was assessed in competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCannabinoid receptor 1(Mus musculus (Mouse))
Jenrin Discovery

US Patent
LigandPNGBDBM286107(US10617673, Example 4a (2S,4'R) | US11179370, Exam...)
Affinity DataIC50:  5.50E+3nMAssay Description:Compound binding to CB1R was assessed in competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCannabinoid receptor 1(Mus musculus (Mouse))
Jenrin Discovery

US Patent
LigandPNGBDBM286101(US10617673, Example 1a (4'R) | US11179370, Example...)
Affinity DataIC50:  5.50E+3nMAssay Description:Compound binding to CB1R was assessed in competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCannabinoid receptor 1(Mus musculus (Mouse))
Jenrin Discovery

US Patent
LigandPNGBDBM286103(US10617673, Example 2a (2S,3R,4'R) | US11179370, E...)
Affinity DataIC50:  5.50E+3nMAssay Description:Compound binding to CB1R was assessed in competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain....More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent