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Found 1 Enz. Inhib. hit(s) for PDB: 1H08
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Astrazeneca

LigandPNGBDBM7627(2,4-bis anilino pyrimidine deriv. 23 | 5-bromo-2-N...)
Affinity DataIC50:  300nMAssay Description:The kinase activity was assayed using an in vitro scintillation proximity assay (SPA) for measuring incorporation of [gamma-33P] ATP into GST-Rb.More data for this Ligand-Target Pair