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Found 1 Enz. Inhib. hit(s) for PDB: 1PYE
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
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LigandPNGBDBM6676(3-benzoyl-6-[(2,6-difluorophenyl)carbonyl]imidazo[...)
Affinity DataIC50:  324nMT: 2°CAssay Description:In vitro CDK assay using purified enzyme, was incubated at room temperature with substrate, and test compounds in the presence of ATP/[gamma-33P]ATP....More data for this Ligand-Target Pair