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Found 2 Enz. Inhib. hit(s) for PDB: 1TFT
TargetE3 ubiquitin-protein ligase XIAP(Homo sapiens (Human))
Queen'S University Of Belfast

Curated by ChEMBL
LigandPNGBDBM13174((2S,4S)-1-[(2S)-3,3-dimethyl-2-[(2S)-2-(methylamin...)
Affinity DataKd:  5nMAssay Description:Binding affinity to XIAP BIR3-domain (unknown origin)More data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase XIAP [241-356](Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM13174((2S,4S)-1-[(2S)-3,3-dimethyl-2-[(2S)-2-(methylamin...)
Affinity DataKd:  5nMpH: 7.4 T: 2°CAssay Description:A fluorescence polarization anisotropy (FPA) competition assay was used to determine the affinities of compounds to BIR3 protein. Fluorescence polari...More data for this Ligand-Target Pair