Compile Data Set for Download or QSAR
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Found 1 Enz. Inhib. hit(s) for PDB: 1V1K
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Astrazeneca

LigandPNGBDBM7599(4,6-bis anilino pyrimidine deriv. 12 | 4-N-{4-[3-(...)
Affinity DataIC50:  3.50E+4nMAssay Description:The kinase activity was assayed using an in vitro scintillation proximity assay (SPA) for measuring incorporation of [gamma-33P] ATP into GST-Rb.More data for this Ligand-Target Pair