Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) for PDB: 2BHE
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Schering

LigandPNGBDBM54680((3Z)-5-bromanyl-3-(3-oxidanylidene-1H-indol-2-ylid...)
Affinity DataIC50:  80nMpH: 8.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Egyptian Russian University

Curated by ChEMBL
LigandPNGBDBM50142632(CHEMBL1231469)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of GST-tagged recombinant human CDK2/cyclin E expressed in insect SF-9 cells after 10 mins by scintillation counting analysis in presence ...More data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Schering

LigandPNGBDBM54680((3Z)-5-bromanyl-3-(3-oxidanylidene-1H-indol-2-ylid...)
Affinity DataIC50:  1.00E+3nMpH: 8.0 T: 2°CAssay Description:Inhibition assay using CDK and selective kinases such as gsk3, EGFR, c-Kit, InsR and KDR.More data for this Ligand-Target Pair