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Found 1 Enz. Inhib. hit(s) for PDB: 2G1Y
TargetRenin(Homo sapiens (Human))
Pfizer

LigandPNGBDBM17982(1,4-benzoxazin-3-one, 19 | 6-(2,4-diamino-6-ethylp...)
Affinity DataIC50:  90nMpH: 7.4 T: 2°CAssay Description:The renin assay utilized a tandem Green Flourescent Protein (tGFP) substrate that was hydrolyzed by human rennin. The tGFP substrate contained a nine...More data for this Ligand-Target Pair