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Found 1 Enz. Inhib. hit(s) for PDB: 2WMW
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
The Institute Of Cancer Research

LigandPNGBDBM33213(pyrazolopyridine, 12)
Affinity DataIC50:  390nMpH: 7.5 T: 2°CAssay Description:CHK kinase function was measured in a DELFIA assay in order to monitor phosphorylation of a CDC25C peptide using a specific phospho antibody. The enz...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB