Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) for PDB: 2WMX
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
The Institute Of Cancer Research

LigandPNGBDBM33217(pyrazolopyridine, (S)-14)
Affinity DataIC50:  860nMpH: 7.5 T: 2°CAssay Description:CHK kinase function was measured in a DELFIA assay in order to monitor phosphorylation of a CDC25C peptide using a specific phospho antibody. The enz...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase Chk1(Homo sapiens (Human))
The Institute Of Cancer Research

LigandPNGBDBM33215(pyrazolopyridine, (Rac)-14 | racemic)
Affinity DataIC50:  890nMpH: 7.5 T: 2°CAssay Description:CHK kinase function was measured in a DELFIA assay in order to monitor phosphorylation of a CDC25C peptide using a specific phospho antibody. The enz...More data for this Ligand-Target Pair