Found 41 Enz. Inhib. hit(s) for PDB: 3LBD 
Affinity DataKi: 0.5nMAssay Description:Binding affinity towards cRARbeta2 receptor by displacing 1.1 nM 3[H]-9-cis-RAMore data for this Ligand-Target Pair
3D Structure (crystal)Affinity DataKi: 0.700nMAssay Description:Binding affinity towards cRARbeta2 receptor by displacing 1.1 nM 3[H]-9-cis-RAMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Agonistic activity of the compound towards retinoic acid receptor-gammaMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Inhibition of [3H]-ATRA binding to Retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Inhibition of [3H]-ATRA binding to Retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Binding affinity against retinoic Acid beta receptor using [3H]- -9-cis-Retinoic Acid in competitive binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Binding affinity against retinoic Acid gamma receptor using [3H]- -9-cis-Retinoic Acid in competitive binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 22nMAssay Description:Effective concentration against Retinoic acid receptor betaMore data for this Ligand-Target Pair
Affinity DataEC50: 12nMAssay Description:Effective concentration against RAR-gamma receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 52nMAssay Description:Transcriptional activation in CV-1 cells expressing Retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Transcriptional activation of Retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
Affinity DataEC50: 45nMAssay Description:Transcriptional activation of Retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
Affinity DataKd: 7nMAssay Description:Dissociation constant for binding to Retinoic acid receptor betaMore data for this Ligand-Target Pair
Affinity DataKd: 17nMAssay Description:Dissociation constant for binding to Retinoic acid receptor gammaMore data for this Ligand-Target Pair
Affinity DataKd: 148nMAssay Description:Inhibition of [3H]-RA binding to retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
Affinity DataKd: 97nMAssay Description:Inhibition of [3H]-RA binding to retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
Affinity DataEC50: 6nMAssay Description:Transcriptional activation of Retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 3.30nMAssay Description:Transcriptional activation of Retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
Affinity DataKd: 100nMAssay Description:Inhibition of [3H]-ATRA binding to baculovirus expressed retinoic acid receptor RAR-betaMore data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 3nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
Affinity DataKd: 150nMAssay Description:Inhibition of [3H]-ATRA binding to baculovirus expressed retinoic acid receptor RAR-gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Transcriptional activation in CV-1 cells expresing human Retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
Affinity DataKd: 0.800nMAssay Description:Dissociation constant for Retinoic acid receptor gammaMore data for this Ligand-Target Pair
Affinity DataKd: 22nMAssay Description:Compound was tested for binding affinity against retinoic acid receptor using 5 nM of [3H]-RA as a radioligand in baculovirus expressed receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 3.30nMAssay Description:Transcriptional activation for RAR beta receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 6nMAssay Description:Transcriptional activation for RAR gamma receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Agonist activity for retinoic acid receptor RAR beta in transcriptional activation assayMore data for this Ligand-Target Pair
Affinity DataEC50: 45nMAssay Description:Agonist activity for retinoic acid receptor RAR gamma in transcriptional activation assayMore data for this Ligand-Target Pair
Affinity DataKd: 97nMAssay Description:Transcriptional activation in CV-1 cells expresing human Retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
Affinity DataKd: 148nMAssay Description:Transcriptional activation in CV-1 cells expresing human Retinoid X receptor RXR-alphaMore data for this Ligand-Target Pair
Affinity DataKd: 7nMAssay Description:Compound was tested for functional activity in CV-1 cells transfected with an expression vector for retinoic acid receptor alpha using transactivatio...More data for this Ligand-Target Pair
Affinity DataEC50: 45nMAssay Description:Compound was tested for functional activity in CV-1 cells transfected with an expression vector for retinoid X receptor alpha using transactivation a...More data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Binding affinity against retinoic Acid beta receptors cotransfected into CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 6nMAssay Description:Transcriptional activation of Retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 3.30nMAssay Description:Transcriptional activation of Retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
Affinity DataEC50: 74nMAssay Description:Transcriptional activation in CV-1 cells expressing Retinoic acid receptor RAR gammaMore data for this Ligand-Target Pair
Affinity DataEC50: 45nMAssay Description:Binding affinity against retinoic Acid gamma receptors cotransfected into CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 29nMAssay Description:Transcriptional activation in CV-1 cells expresing human Retinoic acid receptor RAR betaMore data for this Ligand-Target Pair
Affinity DataKd: 0.800nMpH: 7.9 T: 2°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
Affinity DataEC50: 50nMAssay Description:Compound was tested for functional activity in CV-1 cells transfected with an expression vector for retinoic acid receptor beta using transactivation...More data for this Ligand-Target Pair
