Compile Data Set for Download or QSAR
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Found 4 Enz. Inhib. hit(s) for PDB: 3TJ2
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of Pittsburgh

US Patent
LigandPNGBDBM50014092(CHEMBL3259830 | US9187441, 9l)
Affinity DataKi:  300nM ΔG°:  -36.6kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of Pittsburgh

US Patent
LigandPNGBDBM50014092(CHEMBL3259830 | US9187441, 9l)
Affinity DataKi:  400nMAssay Description:Displacement of fluorescent P4 peptide from MDM2 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of Pittsburgh

US Patent
LigandPNGBDBM50014092(CHEMBL3259830 | US9187441, 9l)
Affinity DataKi:  400nM ΔG°:  -35.9kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
University Of Pittsburgh

US Patent
LigandPNGBDBM50014092(CHEMBL3259830 | US9187441, 9l)
Affinity DataKi:  700nM ΔG°:  -34.5kJ/moleT: 2°CAssay Description:Fluorescent polarization experiments were performed as follows. Briefly, the fluorescence polarization experiments were read on an Ultra Evolution 38...More data for this Ligand-Target Pair