Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) for PDB: 3VSX
TargetRenin(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50387268(CHEMBL2048571)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of human purified reninMore data for this Ligand-Target Pair
TargetRenin(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50387268(CHEMBL2048571)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of human recombinant renin using Arg-Glu(EDANS)-Ile-His-Pro-Phe-His-Leu-Val-Ile-His-Thr-Lys (DABCYL)-Arg as substrate incubated for 10 min...More data for this Ligand-Target Pair
TargetRenin(Macaca fascicularis)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50387268(CHEMBL2048571)
Affinity DataIC50:  7nMAssay Description:Inhibition of renin in cynomolgus monkey plasma after 1 hr by RIAMore data for this Ligand-Target Pair
TargetRenin(Macaca fascicularis)
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50387268(CHEMBL2048571)
Affinity DataIC50:  7nMAssay Description:Inhibition of renin in cynomolgus monkey plasmaMore data for this Ligand-Target Pair