Compile Data Set for Download or QSAR
maximum 50k data
Found 1 Enz. Inhib. hit(s) for PDB: 4G17
TargetCasein kinase I isoform gamma-2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50390498(CHEMBL2071612)
Affinity DataIC50:  1.51E+3nMAssay Description:Inhibition of CK1gamma2 expressed in HEK293 cells assessed as inhibition of LRP6 Thr1479 phosphorylation by immunoblottingMore data for this Ligand-Target Pair