Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) for PDB: 4GHI
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Peloton Therapeutics

Curated by ChEMBL
LigandPNGBDBM50426208(CHEMBL2311933)
Affinity DataIC50:  490nMAssay Description:Binding affinity to His-tagged HIF-2alpha PAS-B domain (unknown origin) after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
TargetEndothelial PAS domain-containing protein 1(Homo sapiens (Human))
Peloton Therapeutics

Curated by ChEMBL
LigandPNGBDBM50426208(CHEMBL2311933)
Affinity DataKd:  90nMAssay Description:Binding affinity to wild type PAS-B domain of HIF-2alpha (unknown origin) by isothermal calorimetry analysisMore data for this Ligand-Target Pair