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Found 3 Enz. Inhib. hit(s) for PDB: 4GU6
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50425675(CHEMBL2315579)
Affinity DataIC50:  195nMAssay Description:Inhibition of FAK (unknown origin) using biotinylated His-TEV-hsFAK(31-686)(K454R) substrate after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50425675(CHEMBL2315579)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of FAK in human HT-29 cells assessed as phosphorylation at tyrosine 397 after 45 minsMore data for this Ligand-Target Pair
TargetFocal adhesion kinase 1(Homo sapiens (Human))
Merck Serono

Curated by ChEMBL
LigandPNGBDBM50425675(CHEMBL2315579)
Affinity DataKd:  44nMAssay Description:Binding affinity to FAK (unknown origin) by surface plasmon resonance analysisMore data for this Ligand-Target Pair