Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) for PDB: 4KKH
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50430432(CHEMBL2334705)
Affinity DataIC50:  1.09E+3nMAssay Description:Inhibition of JNK3 in human SH-SY5Y cells assessed as decrease in anisomycin-induced TNFalpha mRNA level incubated for 1 hr prior to anisomycin induc...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50430432(CHEMBL2334705)
Affinity DataKd:  46nMAssay Description:Binding affinity to N-terminal His6X-tagged human recombinant JNK3 catalytic domain expressed in Escherichia coli BL21 (DE3) by surface plasmon reson...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
Hanyang University

Curated by ChEMBL
LigandPNGBDBM50430432(CHEMBL2334705)
Affinity DataKd:  46nMAssay Description:Binding affinity to JNK3 (unknown origin) by surface plasmon resonance analysis in presence of ATPMore data for this Ligand-Target Pair