Affinity DataIC50: 1.42E+3nMAssay Description:Inhibition of biotin-tagged human GKRP-fluorescein-tagged human GK interaction preincubated for 20 mins followed by fluorescein-tagged human GK addit...More data for this Ligand-Target Pair
Affinity DataKd: 240nMAssay Description:Binding affinity to GKRP (unknown origin) by surface plasmon resonance analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 3.64E+3nMAssay Description:Inhibition of GKRP-GK interaction in rat primary hepatocytes assessed as translocation of GK from nucleus to cytoplasm preincubated for 20 mins follo...More data for this Ligand-Target Pair