Compile Data Set for Download or QSAR
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Found 5 Enz. Inhib. hit(s) for PDB: 4QM0
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50012123(CHEMBL3263696)
Affinity DataIC50:  130nMAssay Description:Displacement of [3H]25-hydroxycholesterol from human RORc-LBD expressed in bacterial expression system after 3 hrs by scintillation counting analysisMore data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50012123(CHEMBL3263696)
Affinity DataIC50:  130nMAssay Description:Displacement of [3H2]25-hydroxycholesterol from human RORc-LBD after 3 hrs by scintillation countingMore data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50012123(CHEMBL3263696)
Affinity DataEC50:  460nMAssay Description:Inverse agonist activity at N-terminal 6xHis-tagged human RORc ligand binding domain expressed in bacterial expression system assessed as inhibition ...More data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50012123(CHEMBL3263696)
Affinity DataEC50:  1.00E+3nMAssay Description:Inverse agonist activity at human GAL4-fused RORc expressed in HEK293 cells after 5 hrs by luciferase reporter gene based transcriptional assayMore data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50012123(CHEMBL3263696)
Affinity DataEC50:  460nMAssay Description:Inverse agonist activity at an N-terminal 6xHis-GST-tag human RORc-LBD assessed as inhibition of recruitment of the SRC1 co-activator peptide after 3...More data for this Ligand-Target Pair