Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) for PDB: 4ZJW
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50108884(CHEMBL3596600)
Affinity DataIC50:  100nMAssay Description:Inverse agonist activity at human recombinant GST-tagged RORgammat ligand binding domain assessed as effect on receptor-biotin tagged TRAP220 co-acti...More data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50108884(CHEMBL3596600)
Affinity DataEC50:  200nMAssay Description:Inverse agonist activity at Gal4 DNA binding domain-tagged human RORgammat expressed in HEK293T cells assessed as effect on receptor-mediated transcr...More data for this Ligand-Target Pair