Compile Data Set for Download or QSAR
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Found 25 Enz. Inhib. hit(s) with all data for entry = 50008567
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074768(2-{2-[Bis-(4-methoxycarbonyl-phenoxy)-phosphoryl]-...)
Affinity DataIC50:  16nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074760(2-(2-{Bis-[4-(ethoxycarbonylmethyl-carbamoyl)-phen...)
Affinity DataIC50:  23nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074762(2-{2-[Bis-(4-propylcarbamoyl-phenoxy)-phosphoryl]-...)
Affinity DataIC50:  30nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074769(2-(2-{Bis-[4-(2-methoxycarbonyl-ethylcarbamoyl)-ph...)
Affinity DataIC50:  36nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074753(2-{2-[Bis-(4-methanesulfonylamino-phenoxy)-phospho...)
Affinity DataIC50:  400nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074766(2-{2-[Bis-(4-acetylamino-phenoxy)-phosphoryl]-pyrr...)
Affinity DataIC50:  400nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074759(2-(2-{Bis-[4-(2-amino-acetylamino)-phenoxy]-phosph...)
Affinity DataIC50:  500nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074770(2-(2-{[4-((R)-2-Amino-propionylamino)-phenoxy]-[4-...)
Affinity DataIC50:  600nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074772(2-(2-{Bis-[4-(2-benzoylamino-acetylamino)-phenoxy]...)
Affinity DataIC50:  700nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074756(2-{2-[Bis-(3-acetylamino-phenoxy)-phosphoryl]-pyrr...)
Affinity DataIC50:  800nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074767(2-(2-{Bis-[4-(2-acetylamino-2-methoxycarbonyl-ethy...)
Affinity DataIC50:  1.40E+3nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074765(2-{2-[(5-Ureido-cyclohexa-1,3-dienyloxy)-(3-ureido...)
Affinity DataIC50:  2.30E+3nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074761((R)-2-[2-(Diphenoxy-phosphoryl)-pyrrolidine-1-carb...)
Affinity DataIC50:  5.00E+3nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074752(2-(2-{Bis-[4-(pyrrolidin-1-ylamino)-phenoxy]-phosp...)
Affinity DataIC50:  5.00E+3nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074758((S)-2-[2-(Diphenoxy-phosphoryl)-pyrrolidine-1-carb...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074757(2-{2-[Bis-(4-methoxy-phenoxy)-phosphoryl]-pyrrolid...)
Affinity DataIC50:  2.20E+4nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074751((S)-2-[2-(6-Oxo-5,7-dioxa-6lambda*5*-phospha-diben...)
Affinity DataIC50:  3.10E+4nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074764((S)-2-{2-[(2'-Hydroxy-biphenyl-2-yloxy)-methoxy-ph...)
Affinity DataIC50:  4.70E+4nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074756(2-{2-[Bis-(3-acetylamino-phenoxy)-phosphoryl]-pyrr...)
Affinity DataIC50:  5.00E+4nMAssay Description:Effect of the compound on the activity of prolyl endopeptidase (PEP) was evaluated at 1 mM concentration for DPP IVMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074761((R)-2-[2-(Diphenoxy-phosphoryl)-pyrrolidine-1-carb...)
Affinity DataIC50:  8.30E+4nMAssay Description:Effect of the compound on the activity of membrane alanyl aminopeptidase (MAAP) is evaluated at at a concentration of 1 mM.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074756(2-{2-[Bis-(3-acetylamino-phenoxy)-phosphoryl]-pyrr...)
Affinity DataIC50:  8.90E+4nMAssay Description:Effect of the compound on the activity of prolyl endopeptidase (PEP) was evaluated at the IC50 concentration for DPP IV andMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAminopeptidase N(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074760(2-(2-{Bis-[4-(ethoxycarbonylmethyl-carbamoyl)-phen...)
Affinity DataIC50:  1.04E+5nMAssay Description:Effect of the compound on the activity of membrane alanyl aminopeptidase (MAAP) is evaluated at the IC50 concentration for DPPIV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074754(2-{2-[Bis-(4-hydroxy-phenoxy)-phosphoryl]-pyrrolid...)
Affinity DataIC50:  1.90E+5nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074763(2-{2-[Bis-(2,2,2-trichloro-ethoxy)-phosphoryl]-pyr...)
Affinity DataIC50:  1.80E+6nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
University Of Antwerp (Uia)

Curated by ChEMBL
LigandPNGBDBM50074755(2-{2-[Bis-(2,2,2-trifluoro-ethoxy)-phosphoryl]-pyr...)
Affinity DataIC50:  9.10E+6nMAssay Description:In vitro inhibition of human Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed