Compile Data Set for Download or QSAR
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Found 31 Enz. Inhib. hit(s) with all data for entry = 50008813
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50077519(1-(2-Fluoro-ethyl)-3-((4Z,7Z,10Z,13Z)-nonadeca-4,7...)
Affinity DataKi:  52nMAssay Description:The compound was tested for Ki value against rat whole brain P2 membrane preparation in absence of enzyme inhibitor PMSFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50077519(1-(2-Fluoro-ethyl)-3-((4Z,7Z,10Z,13Z)-nonadeca-4,7...)
Affinity DataKi:  55nMAssay Description:The compound was tested for Ki value against rat whole brain P2 membrane preparation in presence of enzyme inhibitor PMSF.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM22988((5Z,8Z,11Z,14Z)-N-(2-hydroxyethyl)icosa-5,8,11,14-...)
Affinity DataKi:  89nMAssay Description:The compound was tested for Ki value against rat whole brain P2 membrane preparation in presence of enzyme inhibitor PMSF.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50077510(1-((4Z,7Z,10Z,13Z)-Nonadeca-4,7,10,13-tetraenyl)-3...)
Affinity DataKi:  91nMAssay Description:The compound was tested for Ki value against rat whole brain P2 membrane preparation in presence of enzyme inhibitor PMSF.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50077522(1-Isopropyl-3-((4Z,7Z,10Z,13Z)-nonadeca-4,7,10,13-...)
Affinity DataKi:  131nMAssay Description:The compound was tested for Ki value against rat whole brain P2 membrane preparation in presence of enzyme inhibitor PMSF.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50077511(1-Ethyl-3-((4Z,7Z,10Z,13Z)-nonadeca-4,7,10,13-tetr...)
Affinity DataKi:  156nMAssay Description:The compound was tested for Ki value against rat whole brain P2 membrane preparation in presence of enzyme inhibitor PMSF.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50077510(1-((4Z,7Z,10Z,13Z)-Nonadeca-4,7,10,13-tetraenyl)-3...)
Affinity DataKi:  170nMAssay Description:The compound was tested for Ki value against rat whole brain P2 membrane preparation in absence of enzyme inhibitor PMSFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50077522(1-Isopropyl-3-((4Z,7Z,10Z,13Z)-nonadeca-4,7,10,13-...)
Affinity DataKi:  204nMAssay Description:The compound was tested for Ki value against rat whole brain P2 membrane preparation in absence of enzyme inhibitor PMSFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50077531(((4Z,7Z,10Z,13Z)-Nonadeca-4,7,10,13-tetraenyl)-car...)
Affinity DataKi:  218nMAssay Description:The compound was tested for Ki value against rat whole brain P2 membrane preparation in presence of enzyme inhibitor PMSF.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50077525(((4Z,7Z,10Z,13Z)-Nonadeca-4,7,10,13-tetraenyl)-car...)
Affinity DataKi:  331nMAssay Description:The compound was tested for Ki value against rat whole brain P2 membrane preparation in presence of enzyme inhibitor PMSF.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50077521(1-Isobutyl-3-((4Z,7Z,10Z,13Z)-nonadeca-4,7,10,13-t...)
Affinity DataKi:  335nMAssay Description:The compound was tested for Ki value against rat whole brain P2 membrane preparation in presence of enzyme inhibitor PMSF.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50077516(1-(2-Hydroxy-ethyl)-3-((4Z,7Z,10Z,13Z)-nonadeca-4,...)
Affinity DataKi:  347nMAssay Description:The compound was tested for Ki value against rat whole brain P2 membrane preparation in presence of enzyme inhibitor PMSF.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50077532(1-Methyl-3-((4Z,7Z,10Z,13Z)-nonadeca-4,7,10,13-tet...)
Affinity DataKi:  436nMAssay Description:The compound was tested for Ki value against rat whole brain P2 membrane preparation in presence of enzyme inhibitor PMSF.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50077526(CHEMBL61055 | Propyl-carbamic acid (5Z,8Z,11Z,14Z)...)
Affinity DataKi:  471nMAssay Description:The compound was tested for Ki value against rat whole brain P2 membrane preparation in presence of enzyme inhibitor PMSF.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50077528(CHEMBL61918 | [((5Z,8Z,11Z,14Z)-Icosa-5,8,11,14-te...)
Affinity DataKi:  578nMAssay Description:The compound was tested for Ki value against rat whole brain P2 membrane preparation in presence of enzyme inhibitor PMSF.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50077523(1-(2-Methoxy-ethyl)-3-((4Z,7Z,10Z,13Z)-nonadeca-4,...)
Affinity DataKi:  746nMAssay Description:The compound was tested for Ki value against rat whole brain P2 membrane preparation in presence of enzyme inhibitor PMSF.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50077517(2-[((5Z,8Z,11Z,14Z)-Icosa-5,8,11,14-tetraenyl)oxy]...)
Affinity DataKi:  797nMAssay Description:The compound was tested for Ki value against rat whole brain P2 membrane preparation in presence of enzyme inhibitor PMSF.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50077520((5Z,8Z,11Z,14Z)-1-Isopropoxy-icosa-5,8,11,14-tetra...)
Affinity DataKi:  871nMAssay Description:The compound was tested for Ki value against rat whole brain P2 membrane preparation in presence of enzyme inhibitor PMSF.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50077514((5Z,8Z,11Z,14Z)-1-(2-Fluoro-ethoxy)-icosa-5,8,11,1...)
Affinity DataKi:  885nMAssay Description:The compound was tested for Ki value against rat whole brain P2 membrane preparation in presence of enzyme inhibitor PMSF.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50077529(CHEMBL61107 | Isopropyl-carbamic acid (5Z,8Z,11Z,1...)
Affinity DataKi:  995nMAssay Description:The compound was tested for Ki value against rat whole brain P2 membrane preparation in presence of enzyme inhibitor PMSF.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50077533((5Z,8Z,11Z,14Z)-1-Propoxy-icosa-5,8,11,14-tetraene...)
Affinity DataKi:  1.08E+3nMAssay Description:The compound was tested for Ki value against rat whole brain P2 membrane preparation in presence of enzyme inhibitor PMSF.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50077509((5Z,8Z,11Z,14Z)-1-Allyloxy-icosa-5,8,11,14-tetraen...)
Affinity DataKi:  1.17E+3nMAssay Description:The compound was tested for Ki value against rat whole brain P2 membrane preparation in presence of enzyme inhibitor PMSF.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50077512(((4Z,7Z,10Z,13Z)-Nonadeca-4,7,10,13-tetraenyl)-car...)
Affinity DataKi:  1.23E+3nMAssay Description:The compound was tested for Ki value against rat whole brain P2 membrane preparation in presence of enzyme inhibitor PMSF.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50077530((5Z,8Z,11Z,14Z)-1-sec-Butoxy-icosa-5,8,11,14-tetra...)
Affinity DataKi:  1.31E+3nMAssay Description:The compound was tested for Ki value against rat whole brain P2 membrane preparation in presence of enzyme inhibitor PMSF.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50077527((5Z,8Z,11Z,14Z)-1-Prop-2-ynyloxy-icosa-5,8,11,14-t...)
Affinity DataKi:  1.58E+3nMAssay Description:The compound was tested for Ki value against rat whole brain P2 membrane preparation in presence of enzyme inhibitor PMSF.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50077518((5Z,8Z,11Z,14Z)-1-Butoxy-icosa-5,8,11,14-tetraene ...)
Affinity DataKi:  1.71E+3nMAssay Description:The compound was tested for Ki value against rat whole brain P2 membrane preparation in presence of enzyme inhibitor PMSF.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50077534(CHEMBL294826 | Ethyl-carbamic acid (5Z,8Z,11Z,14Z)...)
Affinity DataKi:  2.20E+3nMAssay Description:The compound was tested for Ki value against rat whole brain P2 membrane preparation in presence of enzyme inhibitor PMSF.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50077524((5Z,8Z,11Z,14Z)-1-Ethoxy-icosa-5,8,11,14-tetraene ...)
Affinity DataKi:  2.20E+3nMAssay Description:The compound was tested for Ki value against rat whole brain P2 membrane preparation in presence of enzyme inhibitor PMSF.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50077513((5Z,8Z,11Z,14Z)-1-Isobutoxy-icosa-5,8,11,14-tetrae...)
Affinity DataKi:  2.48E+3nMAssay Description:The compound was tested for Ki value against rat whole brain P2 membrane preparation in presence of enzyme inhibitor PMSF.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM50077515((5Z,8Z,11Z,14Z)-1-Methoxy-icosa-5,8,11,14-tetraene...)
Affinity DataKi:  4.26E+3nMAssay Description:The compound was tested for Ki value against rat whole brain P2 membrane preparation in presence of enzyme inhibitor PMSF.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Organix

Curated by ChEMBL
LigandPNGBDBM22988((5Z,8Z,11Z,14Z)-N-(2-hydroxyethyl)icosa-5,8,11,14-...)
Affinity DataKi:  5.40E+3nMAssay Description:The compound was tested for Ki value against rat whole brain P2 membrane preparation in absence of enzyme inhibitor PMSFMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed