Compile Data Set for Download or QSAR
maximum 50k data
Found 79 Enz. Inhib. hit(s) with all data for entry = 5225
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM82255(D-Phe-Cys-Tyr-D-Trp-Lys-Abu-Cys-Nal-NH | NC8-12)
Affinity DataKi:  0.0240nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM82460(L-Ser-L-Ala-L-Asn-L-Ser-L-Asn-L-Pro-L-Ala-L-Met-L-...)
Affinity DataKi:  0.0500nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM85521(CAS_5311372 | L-779,976 | NSC_5311372)
Affinity DataKi:  0.0500nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM82255(D-Phe-Cys-Tyr-D-Trp-Lys-Abu-Cys-Nal-NH | NC8-12)
Affinity DataKi:  0.0900nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CAS_38916-34-6 | CB6417646...)
Affinity DataKi:  0.100nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM82460(L-Ser-L-Ala-L-Asn-L-Ser-L-Asn-L-Pro-L-Ala-L-Met-L-...)
Affinity DataKi:  0.100nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM50051568((3S,6S,9S,12R,15S,18S)-9-(4-Amino-butyl)-3-benzyl-...)
Affinity DataKi:  0.100nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM85052(BIM 23197 | BIM-23197)
Affinity DataKi:  0.190nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CAS_38916-34-6 | CB6417646...)
Affinity DataKi:  0.200nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM82460(L-Ser-L-Ala-L-Asn-L-Ser-L-Asn-L-Pro-L-Ala-L-Met-L-...)
Affinity DataKi:  0.200nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CAS_38916-34-6 | CB6417646...)
Affinity DataKi:  0.200nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CAS_38916-34-6 | CB6417646...)
Affinity DataKi:  0.300nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM82460(L-Ser-L-Ala-L-Asn-L-Ser-L-Asn-L-Pro-L-Ala-L-Met-L-...)
Affinity DataKi:  0.300nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM81767(15-28-Somatostatin-28 | CAS_38916-34-6 | CB6417646...)
Affinity DataKi:  0.300nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM82460(L-Ser-L-Ala-L-Asn-L-Ser-L-Asn-L-Pro-L-Ala-L-Met-L-...)
Affinity DataKi:  0.300nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM50063839(BIM 23268 | CHEMBL263606 | H-cyclo[DCys-Phe-Phe-DT...)
Affinity DataKi:  0.370nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM50232821((S)-((S)-2-aminopropyl) 6-amino-2-(2-(2-(naphthale...)
Affinity DataKi:  0.400nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM50059090(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKi:  0.400nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM85246(CST17 | Cortistatin | Cortistatin-17 | L-Asp-L-Arg...)
Affinity DataKi:  0.400nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM50063821(CHEMBL414254 | H-DNal-cyclo[Cys-Tyr-DTrp-Lys-Val-D...)
Affinity DataKi:  0.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM85246(CST17 | Cortistatin | Cortistatin-17 | L-Asp-L-Arg...)
Affinity DataKi:  0.5nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM85246(CST17 | Cortistatin | Cortistatin-17 | L-Asp-L-Arg...)
Affinity DataKi:  0.600nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM50063821(CHEMBL414254 | H-DNal-cyclo[Cys-Tyr-DTrp-Lys-Val-D...)
Affinity DataKi:  0.600nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM85246(CST17 | Cortistatin | Cortistatin-17 | L-Asp-L-Arg...)
Affinity DataKi:  0.600nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM50136767(2-[4-(5,7-Difluoro-2-phenyl-1H-indol-3-yl)-butyryl...)
Affinity DataKi:  0.700nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | RC 160 | Vapreotide)
Affinity DataKi:  0.700nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM85519(L-797,591 | L-797591)
Affinity DataKi:  1.40nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM50051568((3S,6S,9S,12R,15S,18S)-9-(4-Amino-butyl)-3-benzyl-...)
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM85080(CH-275 | CH275 | L-Cys(1)-L-Lys-L-Phe-L-Phe-D-Trp-...)
Affinity DataKi:  3.20nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM50232821((S)-((S)-2-aminopropyl) 6-amino-2-(2-(2-(naphthale...)
Affinity DataKi:  3.30nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM85080(CH-275 | CH275 | L-Cys(1)-L-Lys-L-Phe-L-Phe-D-Trp-...)
Affinity DataKi:  4.30nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM50059090(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKi:  4.40nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | RC 160 | Vapreotide)
Affinity DataKi:  5.40nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM50059090(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKi:  5.60nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM85246(CST17 | Cortistatin | Cortistatin-17 | L-Asp-L-Arg...)
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM85052(BIM 23197 | BIM-23197)
Affinity DataKi:  9.80nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM50063839(BIM 23268 | CHEMBL263606 | H-cyclo[DCys-Phe-Phe-DT...)
Affinity DataKi:  15.1nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM50063839(BIM 23268 | CHEMBL263606 | H-cyclo[DCys-Phe-Phe-DT...)
Affinity DataKi:  16.3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM50063839(BIM 23268 | CHEMBL263606 | H-cyclo[DCys-Phe-Phe-DT...)
Affinity DataKi:  18.4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM85520(CAS_5311373 | L-796,778 | NSC_5311373)
Affinity DataKi:  24nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM85052(BIM 23197 | BIM-23197)
Affinity DataKi:  26.8nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM50051568((3S,6S,9S,12R,15S,18S)-9-(4-Amino-butyl)-3-benzyl-...)
Affinity DataKi:  27nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | RC 160 | Vapreotide)
Affinity DataKi:  31nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM50063821(CHEMBL414254 | H-DNal-cyclo[Cys-Tyr-DTrp-Lys-Val-D...)
Affinity DataKi:  43nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM82464(CAS_71306 | NSC_71306 | RC 160 | Vapreotide)
Affinity DataKi:  45nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM50232821((S)-((S)-2-aminopropyl) 6-amino-2-(2-(2-(naphthale...)
Affinity DataKi:  52nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM50063839(BIM 23268 | CHEMBL263606 | H-cyclo[DCys-Phe-Phe-DT...)
Affinity DataKi:  61.6nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM50232821((S)-((S)-2-aminopropyl) 6-amino-2-(2-(2-(naphthale...)
Affinity DataKi:  64nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM50063821(CHEMBL414254 | H-DNal-cyclo[Cys-Tyr-DTrp-Lys-Val-D...)
Affinity DataKi:  66nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Royal Victoria Hospital

Curated by PDSP Ki Database
LigandPNGBDBM50232821((S)-((S)-2-aminopropyl) 6-amino-2-(2-(2-(naphthale...)
Affinity DataKi:  82nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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