Compile Data Set for Download or QSAR
maximum 50k data
Found 10 Enz. Inhib. hit(s) with all data for entry = 50035010
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50080105((3-(1,1-Dimethyl-heptyl)-9-hydroxymethyl-6,6-dimet...)
Affinity DataKi:  0.820nMAssay Description:Ability to displace [3H]-SR- 141716A binding to human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50072775(2-((1R,2R,5R)-5-hydroxy-2-(3-hydroxypropyl)cyclohe...)
Affinity DataKi:  5.20nMAssay Description:Ability to displace [3H]-SR- 141716A binding to human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataKi:  8.90nMAssay Description:Ability to displace [3H]-SR- 141716A binding to human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCannabinoid receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50080103(5,5-Bis-(4-bromo-phenyl)-3-(2-morpholin-4-yl-ethyl...)
Affinity DataKi:  70nMAssay Description:Ability to displace [3H]-SR- 141716A binding to CB1 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50080102(CHEMBL71810 | JWH-030 | Naphthalen-1-yl-(1-pentyl-...)
Affinity DataKi:  87nMAssay Description:Binding affinity for brain CBI receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50080104(5,5-Bis-(4-bromo-phenyl)-3-heptyl-imidazolidine-2,...)
Affinity DataKi:  98nMAssay Description:Ability to displace [3H]-SR- 141716A binding to CB1 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50080106(5,5-Bis-(4-bromo-phenyl)-3-(3-hydroxy-propyl)-imid...)
Affinity DataKi:  103nMAssay Description:Ability to displace [3H]-SR- 141716A binding to CB1 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM21281((11R)-2-methyl-11-(morpholin-4-ylmethyl)-3-(naphth...)
Affinity DataKi:  152nMAssay Description:Ability to displace [3H]-SR- 141716A binding to human CB1 receptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50072775(2-((1R,2R,5R)-5-hydroxy-2-(3-hydroxypropyl)cyclohe...)
Affinity DataIC50:  14nMAssay Description:Ability to displace [3H]-SR- 141716A binding to human CB1 receptor expressed in CHO cell membranes in absence of agonist 5''-guanylyimidodiphosphateMore data for this Ligand-Target Pair
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50072775(2-((1R,2R,5R)-5-hydroxy-2-(3-hydroxypropyl)cyclohe...)
Affinity DataIC50:  28nMAssay Description:Ability to displace [3H]-SR- 141716A binding to human CB1 receptor expressed in CHO cell membranes in presence of agonist 5'-guanylyimidodiphosphate ...More data for this Ligand-Target Pair