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Found 16 Enz. Inhib. hit(s) with all data for entry = 50009169
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50080842(3,6-Bis[3-(4-methylpiperidino)propionamido]acridin...)
Affinity DataIC50:  1.35E+3nMAssay Description:Ability to inhibit human telomerase in a modified cell-free TRAP assay using extracts from A2780 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50080848(3-(2-Methyl-piperidin-1-yl)-N-{6-[3-(2-methyl-pipe...)
Affinity DataIC50:  2.60E+3nMAssay Description:Ability to inhibit human telomerase in a modified cell-free TRAP assay using extracts from A2780 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50080837(3-(2-Ethyl-piperidin-1-yl)-N-{6-[3-(2-ethyl-piperi...)
Affinity DataIC50:  2.70E+3nMAssay Description:Ability to inhibit human telomerase in a modified cell-free TRAP assay using extracts from A2780 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50080847(3,6-Bis(3-piperidinopropionamido)acridine | 3-Pipe...)
Affinity DataIC50:  2.80E+3nMAssay Description:Ability to inhibit human telomerase in a modified cell-free TRAP assay using extracts from A2780 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50080840(3,6-Bis[3-(azepan-1-yl)propionamido]acridine | 3,6...)
Affinity DataIC50:  3.10E+3nMAssay Description:Ability to inhibit human telomerase in a modified cell-free TRAP assay using extracts from A2780 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50080850(3-[2-(2-Hydroxy-ethyl)-piperidin-1-yl]-N-(6-{3-[2-...)
Affinity DataIC50:  4.10E+3nMAssay Description:Ability to inhibit human telomerase in a modified cell-free TRAP assay using extracts from A2780 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50080839(3-(3-Methyl-piperidin-1-yl)-N-{6-[3-(3-methyl-pipe...)
Affinity DataIC50:  4.40E+3nMAssay Description:Ability to inhibit human telomerase in a modified cell-free TRAP assay using extracts from A2780 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50080849(3,6-Bis(3-pyrrolidinopropionamido)acridine | 3-PYR...)
Affinity DataIC50:  5.20E+3nMAssay Description:Ability to inhibit human telomerase in a modified cell-free TRAP assay using extracts from A2780 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50080841(3-(2-Hydroxymethyl-piperidin-1-yl)-N-{6-[3-(2-hydr...)
Affinity DataIC50:  5.40E+3nMAssay Description:Ability to inhibit human telomerase in a modified cell-free TRAP assay using extracts from A2780 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50080844(3-Diethylamino-N-[6-(3-diethylamino-propionylamino...)
Affinity DataIC50:  5.80E+3nMAssay Description:Ability to inhibit human telomerase in a modified cell-free TRAP assay using extracts from A2780 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50080845(3-(4-Hydroxy-piperidin-1-yl)-N-{6-[3-(4-hydroxy-pi...)
Affinity DataIC50:  8.00E+3nMAssay Description:Ability to inhibit human telomerase in a modified cell-free TRAP assay using extracts from A2780 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50080851(3-Dimethylamino-N-[6-(3-dimethylamino-propionylami...)
Affinity DataIC50:  8.20E+3nMAssay Description:Ability to inhibit human telomerase in a modified cell-free TRAP assay using extracts from A2780 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50080852(3,6-Bis[3-(heptamethyleneimino)piperizinopropionam...)
Affinity DataIC50: >5.00E+4nMAssay Description:Ability to inhibit human telomerase in a modified cell-free TRAP assay using extracts from A2780 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50080843(3,6-Bis[(3-morpholinopropionamido)] acridine | 3-M...)
Affinity DataIC50: >5.00E+4nMAssay Description:Ability to inhibit human telomerase in a modified cell-free TRAP assay using extracts from A2780 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50080838(3-(4-Benzyl-piperidin-1-yl)-N-{6-[3-(4-benzyl-pipe...)
Affinity DataIC50: >5.00E+4nMAssay Description:Ability to inhibit human telomerase in a modified cell-free TRAP assay using extracts from A2780 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
The Institute Of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50080846(3,6-Bis[3-(1,3,3-trimethyl-6-azabicyclo[3.2.1]octa...)
Affinity DataIC50: >5.00E+4nMAssay Description:Ability to inhibit human telomerase in a modified cell-free TRAP assay using extracts from A2780 cell lineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed