Compile Data Set for Download or QSAR
maximum 50k data
Found 58 Enz. Inhib. hit(s) with all data for entry = 50009175
TargetProthrombin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080924(CHEMBL83260 | N-[(S)-1-(1-Carbamimidoyl-piperidin-...)
Affinity DataKi:  1.20nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080911(2-((S)-4-Benzyl-2-naphthalen-2-ylmethyl-3,6-dioxo-...)
Affinity DataKi:  3.5nMAssay Description:Inhibitory concentration of the compound required against thrombin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080920(CHEMBL313769 | N-[(S)-1-(1-Carbamimidoyl-piperidin...)
Affinity DataKi:  8nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080916(CHEMBL84084 | N-[(S)-1-(1-Carbamimidoyl-piperidin-...)
Affinity DataKi:  20nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080915(2-((R)-2-Benzyl-4-butyl-3,6-dioxo-piperazin-1-yl)-...)
Affinity DataKi:  32nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080930(2-[(R)-2-Benzyl-3,6-dioxo-4-(3-phenyl-propyl)-pipe...)
Affinity DataKi:  55nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080913((S)-2-{2-[(R)-2-Benzyl-3,6-dioxo-4-(3-phenyl-propy...)
Affinity DataKi:  55nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080918(CHEMBL408553 | N-[(S)-1-(1-Carbamimidoyl-piperidin...)
Affinity DataKi:  55nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080917(CHEMBL83001 | N-[(S)-2-Benzothiazol-2-yl-1-(1-carb...)
Affinity DataKi:  80nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080914(2-[(R)-2-Benzyl-3,6-dioxo-4-(3-phenyl-propyl)-pipe...)
Affinity DataKi:  130nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080912(2-[(R)-2-Benzyl-3,6-dioxo-4-(3-phenyl-propyl)-pipe...)
Affinity DataKi:  825nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080924(CHEMBL83260 | N-[(S)-1-(1-Carbamimidoyl-piperidin-...)
Affinity DataIC50:  18nMAssay Description:Inhibitory concentration of the compound required against thrombin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080920(CHEMBL313769 | N-[(S)-1-(1-Carbamimidoyl-piperidin...)
Affinity DataIC50:  80nMAssay Description:Inhibitory concentration of the compound required against thrombin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080929(2-((R)-2-benzyl-3,6-dioxo-4-(3-phenylpropyl)pipera...)
Affinity DataIC50:  96nMAssay Description:Inhibitory concentration of the compound required against trypsin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080926(2-{(R)-2-Benzyl-4-[3-(4-chloro-phenyl)-propyl]-3,6...)
Affinity DataIC50:  110nMAssay Description:Inhibitory concentration of the compound required against thrombin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080917(CHEMBL83001 | N-[(S)-2-Benzothiazol-2-yl-1-(1-carb...)
Affinity DataIC50:  150nMAssay Description:Inhibitory concentration of the compound required against thrombin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080918(CHEMBL408553 | N-[(S)-1-(1-Carbamimidoyl-piperidin...)
Affinity DataIC50:  160nMAssay Description:Inhibitory concentration of the compound required against thrombin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080921(2-{(R)-2-Benzyl-4-[3-(4-methoxy-phenyl)-propyl]-3,...)
Affinity DataIC50:  160nMAssay Description:Inhibitory concentration of the compound required against thrombin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080930(2-[(R)-2-Benzyl-3,6-dioxo-4-(3-phenyl-propyl)-pipe...)
Affinity DataIC50:  170nMAssay Description:Inhibitory concentration of the compound required against thrombin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080911(2-((S)-4-Benzyl-2-naphthalen-2-ylmethyl-3,6-dioxo-...)
Affinity DataIC50:  170nMAssay Description:Inhibitory concentration of the compound required against thrombin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080923(2-[(R)-2-Benzyl-3,6-dioxo-4-(3-p-tolyl-propyl)-pip...)
Affinity DataIC50:  210nMAssay Description:Inhibitory concentration of the compound required against thrombin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080922(2-{(R)-2-Benzyl-4-[3-(4-nitro-phenyl)-propyl]-3,6-...)
Affinity DataIC50:  210nMAssay Description:Inhibitory concentration of the compound required against thrombin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080919(2-{(R)-2-Benzyl-4-[3-(4-hydroxy-phenyl)-propyl]-3,...)
Affinity DataIC50:  240nMAssay Description:Inhibitory concentration of the compound required against thrombin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080927(2-{(R)-2-Benzyl-4-[3-(3,4-dichloro-phenyl)-propyl]...)
Affinity DataIC50:  250nMAssay Description:Inhibitory concentration of the compound required against thrombin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080933(CHEMBL83692 | N-[(S)-1-(1-Carbamimidoyl-piperidin-...)
Affinity DataIC50:  280nMAssay Description:Inhibitory concentration of the compound required against thrombin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080925(CHEMBL256219 | N-[(S)-1-(1-Carbamimidoyl-piperidin...)
Affinity DataIC50:  340nMAssay Description:Inhibitory concentration of the compound required against trypsin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080915(2-((R)-2-Benzyl-4-butyl-3,6-dioxo-piperazin-1-yl)-...)
Affinity DataIC50:  340nMAssay Description:Inhibitory concentration of the compound required against thrombin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080934(2-[(R)-2-Benzhydryl-3,6-dioxo-4-(3-phenyl-propyl)-...)
Affinity DataIC50:  350nMAssay Description:Inhibitory concentration of the compound required against thrombin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080932(2-{(R)-2-Benzyl-4-[3-(4-isopropyl-phenyl)-propyl]-...)
Affinity DataIC50:  370nMAssay Description:Inhibitory concentration of the compound required against thrombin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080916(CHEMBL84084 | N-[(S)-1-(1-Carbamimidoyl-piperidin-...)
Affinity DataIC50:  390nMAssay Description:Inhibitory concentration of the compound required against thrombin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080913((S)-2-{2-[(R)-2-Benzyl-3,6-dioxo-4-(3-phenyl-propy...)
Affinity DataIC50:  440nMAssay Description:Inhibition of thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080914(2-[(R)-2-Benzyl-3,6-dioxo-4-(3-phenyl-propyl)-pipe...)
Affinity DataIC50:  660nMAssay Description:Inhibitory concentration of the compound required against thrombin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080925(CHEMBL256219 | N-[(S)-1-(1-Carbamimidoyl-piperidin...)
Affinity DataIC50:  880nMAssay Description:Inhibitory concentration of the compound required against thrombin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080928(2-((R)-2-Benzyl-3,6-dioxo-4-phenethyl-piperazin-1-...)
Affinity DataIC50:  990nMAssay Description:Inhibitory concentration of the compound required against thrombin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080931(CHEMBL84083 | N-[(S)-1-(1-Carbamimidoyl-piperidin-...)
Affinity DataIC50:  1.23E+3nMAssay Description:Inhibitory concentration of the compound required against thrombin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080913((S)-2-{2-[(R)-2-Benzyl-3,6-dioxo-4-(3-phenyl-propy...)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibitory concentration of the compound required against trypsin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080929(2-((R)-2-benzyl-3,6-dioxo-4-(3-phenylpropyl)pipera...)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibitory concentration of the compound required against thrombin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080917(CHEMBL83001 | N-[(S)-2-Benzothiazol-2-yl-1-(1-carb...)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibitory concentration of the compound required against trypsin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080923(2-[(R)-2-Benzyl-3,6-dioxo-4-(3-p-tolyl-propyl)-pip...)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibitory concentration of the compound required against trypsin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080916(CHEMBL84084 | N-[(S)-1-(1-Carbamimidoyl-piperidin-...)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibitory concentration of the compound required against trypsin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080926(2-{(R)-2-Benzyl-4-[3-(4-chloro-phenyl)-propyl]-3,6...)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibitory concentration of the compound required against trypsin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080912(2-[(R)-2-Benzyl-3,6-dioxo-4-(3-phenyl-propyl)-pipe...)
Affinity DataIC50:  6.60E+3nMAssay Description:Inhibitory concentration of the compound required against thrombin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080932(2-{(R)-2-Benzyl-4-[3-(4-isopropyl-phenyl)-propyl]-...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibitory concentration of the compound required against trypsin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080927(2-{(R)-2-Benzyl-4-[3-(3,4-dichloro-phenyl)-propyl]...)
Affinity DataIC50:  7.20E+3nMAssay Description:Inhibitory concentration of the compound required against trypsin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080920(CHEMBL313769 | N-[(S)-1-(1-Carbamimidoyl-piperidin...)
Affinity DataIC50:  7.80E+3nMAssay Description:Inhibitory concentration of the compound required against trypsin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080934(2-[(R)-2-Benzhydryl-3,6-dioxo-4-(3-phenyl-propyl)-...)
Affinity DataIC50:  8.50E+3nMAssay Description:Inhibitory concentration of the compound required against trypsin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080914(2-[(R)-2-Benzyl-3,6-dioxo-4-(3-phenyl-propyl)-pipe...)
Affinity DataIC50:  8.70E+3nMAssay Description:Inhibitory concentration of the compound required against trypsin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080922(2-{(R)-2-Benzyl-4-[3-(4-nitro-phenyl)-propyl]-3,6-...)
Affinity DataIC50:  9.10E+3nMAssay Description:Inhibitory concentration of the compound required against trypsin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080930(2-[(R)-2-Benzyl-3,6-dioxo-4-(3-phenyl-propyl)-pipe...)
Affinity DataIC50:  9.10E+3nMAssay Description:Inhibitory concentration of the compound required against trypsin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50080924(CHEMBL83260 | N-[(S)-1-(1-Carbamimidoyl-piperidin-...)
Affinity DataIC50:  9.70E+3nMAssay Description:Inhibitory concentration of the compound required against trypsin was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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