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Found 14 Enz. Inhib. hit(s) with all data for entry = 50036754
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research

Curated by ChEMBL
LigandPNGBDBM50081229(10-(tert-butyl)-2,6-dimethyl-(6E,10Z)-2,6,10-dodec...)
Affinity DataIC50:  31nMAssay Description:Inhibition of recombinant farnesyltransferase (mFTase) in scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research

Curated by ChEMBL
LigandPNGBDBM50081234(3-[(Z)-ethylidene]-7,11-dimethyl-(6E)-1,6,10-dodec...)
Affinity DataIC50:  173nMAssay Description:Inhibition of recombinant farnesyltransferase (mFTase) in scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research

Curated by ChEMBL
LigandPNGBDBM50081235(3-substituted farnesyl diphosphate analogue | 4-[(...)
Affinity DataIC50:  189nMAssay Description:Inhibition of recombinant farnesyltransferase (mFTase) in scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research

Curated by ChEMBL
LigandPNGBDBM50081227(10-ethyl-2,6-dimethyl-(6E,10E)-2,6,10-dodecatriene...)
Affinity DataIC50:  215nMAssay Description:Inhibition of recombinant farnesyltransferase (mFTase) in scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research

Curated by ChEMBL
LigandPNGBDBM50081226(1-[1-[(Z)-ethylidene]-5,9-dimethyl-(4E)-4,8-decadi...)
Affinity DataIC50:  299nMAssay Description:Inhibition of recombinant farnesyltransferase (mFTase) in scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research

Curated by ChEMBL
LigandPNGBDBM50081238(4-[(Z)-ethylidene]-8,12,16-trimethyl-(7E,11E)-1,7,...)
Affinity DataIC50:  453nMAssay Description:Inhibition of recombinant farnesyltransferase (mFTase) in scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Parke-Davis Pharmaceutical Research

Curated by ChEMBL
LigandPNGBDBM50081233(3-[(Z)-ethylidene]-7,11,15-trimethyl-(6E,10E)-1,6,...)
Affinity DataIC50:  715nMAssay Description:Inhibition of recombinant farnesyltransferase (mFTase) in scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50081233(3-[(Z)-ethylidene]-7,11,15-trimethyl-(6E,10E)-1,6,...)
Affinity DataIC50:  3.05E+3nMAssay Description:Inhibition of recombinant Geranylgeranyl transferase type I in scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50081238(4-[(Z)-ethylidene]-8,12,16-trimethyl-(7E,11E)-1,7,...)
Affinity DataIC50:  3.38E+3nMAssay Description:Inhibition of recombinant Geranylgeranyl transferase type I in scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50081229(10-(tert-butyl)-2,6-dimethyl-(6E,10Z)-2,6,10-dodec...)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of recombinant Geranylgeranyl transferase type I in scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50081227(10-ethyl-2,6-dimethyl-(6E,10E)-2,6,10-dodecatriene...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant Geranylgeranyl transferase type I in scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50081234(3-[(Z)-ethylidene]-7,11-dimethyl-(6E)-1,6,10-dodec...)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of recombinant Geranylgeranyl transferase type I in scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50081226(1-[1-[(Z)-ethylidene]-5,9-dimethyl-(4E)-4,8-decadi...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant Geranylgeranyl transferase type I in scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50081235(3-substituted farnesyl diphosphate analogue | 4-[(...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant Geranylgeranyl transferase type I in scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed